SCHEMBL8230677

SCHEMBL8230677

COCCCn1c(NC(=O)c2cccc(N)c2)nc2ccc(C(=O)N3CCOCC3)cc21

nearest known ligand 0.68

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 13/20 0.68
ITK Q08881 1/20 0.51
OPRK1 P41145 2/20 0.47
IRAK4 Q9NWZ3 2/20 0.46
MTOR P42345 1/20 0.46
IRAK1 P51617 1/20 0.46
KDM4E B2RXH2 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8230504 0.94 ADORA2A (0.68) ADORA2AITK
SCHEMBL8230880 0.93 ADORA2A (0.75) ADORA2AITKOPRK1IRAK4
SCHEMBL8230877 0.92 ADORA2A (0.79) ADORA2AITKOPRK1IRAK4
SCHEMBL1468392 0.89 ADORA2A (0.85) ADORA2AITKOPRK1
SCHEMBL8239545 0.86 ADORA2A (0.61) ADORA2AITK
SCHEMBL8247059 0.86 ADORA2A (0.81) ADORA2A
SCHEMBL8233532 0.85 ADORA2A (0.65) ADORA2AITKOPRK1
SCHEMBL8230882 0.85 ADORA2A (0.65) ADORA2AITKOPRK1
SCHEMBL8233912 0.85 ADORA2A (0.79) ADORA2AITKOPRK1
SCHEMBL8240280 0.83 ADORA2A (0.76) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007133983-A2 2-AMINOBENZIMIDAZOLES FOR TREATING NEURODEGENERATIVE DISEASES PHARMACOPEIA, INC. (US) 2007-11-22 WO disclosed