SCHEMBL8230880

SCHEMBL8230880

COCCCn1c(NC(=O)c2cccc(N)c2)nc2ccc(C(=O)N3CCC3)cc21

nearest known ligand 0.75

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 13/20 0.75
OPRK1 P41145 2/20 0.49
CNR2 P34972 1/20 0.48
ITK Q08881 2/20 0.47
IRAK4 Q9NWZ3 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8230877 0.97 ADORA2A (0.79) ADORA2AOPRK1CNR2ITKIRAK4
SCHEMBL8230677 0.93 ADORA2A (0.68) ADORA2AOPRK1ITKIRAK4
SCHEMBL8233912 0.91 ADORA2A (0.79) ADORA2AOPRK1CNR2ITK
SCHEMBL8230882 0.91 ADORA2A (0.65) ADORA2AOPRK1ITK
SCHEMBL8233532 0.91 ADORA2A (0.65) ADORA2AOPRK1ITK
SCHEMBL1468271 0.88 ADORA2A (0.95) ADORA2AOPRK1ITK
SCHEMBL12744804 0.86 ADORA2A (1.00) ADORA2AOPRK1ITK
SCHEMBL8230504 0.86 ADORA2A (0.68) ADORA2AITK
SCHEMBL8246362 0.86 ADORA2A (0.57) ADORA2A
SCHEMBL8247595 0.85 ADORA2A (0.76) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007133983-A2 2-AMINOBENZIMIDAZOLES FOR TREATING NEURODEGENERATIVE DISEASES PHARMACOPEIA, INC. (US) 2007-11-22 WO disclosed