SCHEMBL8234091

SCHEMBL8234091

Cc1ccc2c(c1)nc(C(F)(F)F)n2-c1cnc(NCc2ccncc2C)cn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.35
CYP3A4 P08684 3/20 0.34
RXRA P19793 1/20 0.32
AOC3 Q16853 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
STIM1 Q13586 1/20 0.31
ORAI1 Q96D31 1/20 0.31
KDM4C Q9H3R0 1/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
CYP2C19 P33261 2/20 0.30
LMNA P02545 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
TSHR P16473 1/20 0.30
KCNH2 Q12809 1/20 0.30
HCRTR1 O43613 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL646734 0.89 MAPT (0.36) PDE10ACYP3A4KDM4EALDH1A1STIM1
SCHEMBL11940271 0.89 PTGS2 (0.38) PDE10ACYP3A4RXRAHPGDSTIM1
SCHEMBL646474 0.86 RXRA (0.39) RXRAKDM4EALDH1A1MEN1KMT2A
SCHEMBL647042 0.84 MAPT (0.38) PDE10ACYP3A4KDM4EALDH1A1STIM1
SCHEMBL646334 0.80 MAPT (0.36) PDE10ACYP3A4KDM4EALDH1A1STIM1
SCHEMBL647141 0.78 TSHR (0.38) CYP3A4ALDH1A1HPGDMEN1KMT2A
SCHEMBL646799 0.78 NAMPT (0.37) RXRAKDM4E
SCHEMBL8228712 0.77 MEN1 (0.39) AOC3MEN1KMT2AHCRTR1
SCHEMBL648068 0.76 MKNK1 (0.38) CYP3A4KDM4EALDH1A1CYP2C19CYP1A2
SCHEMBL646764 0.76 ABL1 (0.42) RXRAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007109362-A2 BENZOIMIDAZOLYL-PARAZINE COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES SYNTA PHARMACEUTICALS CORP. (US) 2007-09-27 WO disclosed