SCHEMBL8237644

SCHEMBL8237644

Cc1cc2c(cc1I)OC(F)(F)O2

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
STIM1 Q13586 2/20 0.33
ORAI1 Q96D31 2/20 0.33
GPR3 P46089 1/20 0.33
TSHR P16473 1/20 0.32
CTNNB1 P35222 1/20 0.30
WNT3A P56704 1/20 0.30
SCN9A Q15858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8239476 0.84 TSHR (0.39) STIM1ORAI1GPR3TSHRCTNNB1
SCHEMBL13367746 0.76 STIM1 (0.40) STIM1ORAI1GPR3TSHRCTNNB1
SCHEMBL16044114 0.76 GPR3 (0.34) GPR3CTNNB1WNT3A
SCHEMBL8236665 0.74 CD44 (0.43) STIM1ORAI1GPR3TSHR
SCHEMBL1702518 0.74 STIM1 (0.33) STIM1ORAI1GPR3TSHRCTNNB1
SCHEMBL12279630 0.74 STIM1 (0.33) STIM1ORAI1GPR3TSHRCTNNB1
SCHEMBL31457665 0.74 AHR (0.33) GPR3CTNNB1WNT3A
SCHEMBL1859168 0.74 GPR3 (0.33) GPR3CTNNB1WNT3A
SCHEMBL16076086 0.74 TSHR (0.42) STIM1ORAI1GPR3TSHR
SCHEMBL16044169 0.74 ATP4A (0.36) GPR3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007089034-A1 BENZOXAZINES AND RELATED NITROGEN-CONTAINING HETEROBICYCLIC COMPOUNDS USEFUL AS MINERALOCORTICOID RECEPTOR MODULATING AGENTS MITSUBISHI TANABE PHARMA CORPORATION (JP) 2007-08-09 WO disclosed