SCHEMBL8240207

SCHEMBL8240207

CC(C)(C)c1ccc(C(C(O)CO)N2CCNCC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 7/20 0.46
HPGD P15428 1/20 0.43
LMNA P02545 2/20 0.41
TACR1 P25103 2/20 0.39
RECQL P46063 1/20 0.36
OPRM1 P35372 2/20 0.36
CYP2D6 P10635 1/20 0.36
CYP19A1 P11511 1/20 0.36
HTR1A P08908 1/20 0.35
HTR3A P46098 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8963892 0.76 OPRD1 (0.68) OPRD1HPGDLMNAOPRM1CYP2D6
SCHEMBL12896029 0.72 OGA (0.48) MEN1KMT2A
SCHEMBL12896031 0.70 HDAC1 (0.54)
SCHEMBL11775241 0.68 MEN1 (0.53) OPRD1CYP2D6MEN1KMT2A
SCHEMBL23188717 0.66 LMNA (0.51) LMNATACR1RECQLOPRM1CYP2D6
SCHEMBL31376561 0.66 LMNA (0.51) LMNATACR1RECQLOPRM1CYP2D6
SCHEMBL1629743 0.66 LMNA (0.51) LMNATACR1RECQLOPRM1CYP2D6
SCHEMBL27407639 0.65 CYP3A4 (0.47) LMNACYP2D6MEN1KMT2A
SCHEMBL12473965 0.65 MEN1 (0.58) OPRD1CYP2D6MEN1KMT2A
SCHEMBL15186926 0.64 OPRD1 (0.49) OPRD1TACR1OPRM1CYP2D6CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007082880-A1 PYRIDINE AND PYRIMIDINE DERIVATIVES AS INHIBITORS OF HISTONE DEACETYLASE JANSSEN PHARMACEUTICA N.V. (BE) 2007-07-26 WO disclosed