SCHEMBL8243715

SCHEMBL8243715

O=C(COc1ccc(F)c(Cl)c1)N1CCC(S(=O)(=O)NC2=CCCC=C2)C1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ATF4 P18848 4/20 0.40
RAB9A P51151 3/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
GAA P10253 1/20 0.38
LMNA P02545 2/20 0.37
CPT2 P23786 1/20 0.36
CPT1A P50416 1/20 0.36
CPT1B Q92523 1/20 0.36
NPC1 O15118 2/20 0.36
HTT P42858 1/20 0.36
AOC2 O75106 1/20 0.36
FKBP1A P62942 1/20 0.36
PKM P14618 1/20 0.36
MCHR1 Q99705 1/20 0.36
EPHX2 P34913 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL65663 0.84 ALDH1A1 (0.46) SMN1; SMN2L3MBTL1ATF4RAB9AALDH1A1
SCHEMBL57050 0.79 KMT2A (0.47) SMN1; SMN2L3MBTL1ATF4RAB9AALDH1A1
SCHEMBL66069 0.79 TDP1 (0.47) SMN1; SMN2L3MBTL1ATF4RAB9AALDH1A1
SCHEMBL66545 0.78 ALDH1A1 (0.48) SMN1; SMN2L3MBTL1ATF4RAB9AALDH1A1
SCHEMBL56480 0.78 SMN1; SMN2 (0.53) SMN1; SMN2L3MBTL1ATF4RAB9AALDH1A1
SCHEMBL8243869 0.78 SMN1; SMN2 (0.43) SMN1; SMN2L3MBTL1ATF4RAB9AALDH1A1
SCHEMBL65760 0.74 SMN1; SMN2 (0.50) SMN1; SMN2L3MBTL1ATF4RAB9AALDH1A1
SCHEMBL56987 0.73 KMT2A (0.51) SMN1; SMN2L3MBTL1ATF4ALDH1A1GAA
SCHEMBL8236980 0.67 ALDH1A1 (0.51) SMN1; SMN2L3MBTL1RAB9AALDH1A1MAPT
SCHEMBL19702678 0.65 SMN1; SMN2 (0.44) SMN1; SMN2L3MBTL1ATF4RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007050522-A1 DERIVATIVES FOR MODULATION OF ION CHANNELS VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-05-03 WO disclosed