SCHEMBL824637

SCHEMBL824637

N#Cc1cnn(-c2ncccn2)c1N

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.54
KDM4E B2RXH2 3/20 0.54
MEN1 O00255 1/20 0.54
XDH P47989 2/20 0.49
CDK2 P24941 1/20 0.46
ABL1 P00519 1/20 0.42
KDR P35968 1/20 0.42
ALDH1A1 P00352 3/20 0.42
HPGD P15428 1/20 0.42
NPSR1 Q6W5P4 2/20 0.41
KDM4D Q6B0I6 1/20 0.41
MAPT P10636 2/20 0.40
HTT P42858 1/20 0.40
PKM P14618 1/20 0.40
RXFP1 Q9HBX9 2/20 0.38
GLA P06280 1/20 0.38
PLAUR Q03405 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12017340 0.84 KMT2A (0.53) KMT2AKDM4EMEN1XDHABL1
SCHEMBL824888 0.82 PLAUR (0.52) KMT2AKDM4EMEN1XDHCDK2
SCHEMBL12062825 0.81 CDK2 (0.42) KMT2AKDM4EMEN1XDHCDK2
SCHEMBL18751770 0.80 CDK2 (0.45) KMT2AKDM4EMEN1CDK2ALDH1A1
SCHEMBL840161 0.78 KMT2A (0.53) KMT2AKDM4EMEN1XDHCDK2
SCHEMBL839931 0.78 KMT2A (0.53) KMT2AKDM4EMEN1XDHCDK2
SCHEMBL839641 0.78 KMT2A (0.48) KMT2AKDM4EMEN1XDHCDK2
SCHEMBL13430466 0.76 KMT2A (0.53) KMT2AKDM4EMEN1XDHABL1
SCHEMBL60939 0.76 KMT2A (0.71) KMT2AKDM4EMEN1XDHALDH1A1
SCHEMBL12945645 0.76 KDM4E (0.49) KMT2AKDM4EMEN1XDHCDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 43 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2253672-B1 AZO PIGMENTS AND DISPERSION, COLORING COMPOSITION AND INK FOR INK-JET RECORDING CONTAINING THE AZO PIGMENTS, INK-JET RECORDING METHOD AND RECORDED PRODUCT FUJIFILM CORP (JP) 2016-11-23 EP disclosed
EP-2319890-B1 AZO COMPOUND, AZO PIGMENT, PIGMENT DISPERSION, COLOR COMPOSITION, INKJET RECORDING INK, COLOR COMPOSITION FOR COLOR FILTER, COLOR FILTER, AND METHOD FOR PREPARING COLOR COMPOSITION FOR COLOR FILTER FUJIFILM CORP (JP) 2015-10-28 EP disclosed
US-8828132-B2 Pigment composition, ink for inkjet recording, coloring composition for color filter, and color filter FUJIFILM CORPORATION (JP) 2014-09-09 US disclosed
US-8470054-B2 Azo compound, azo pigment, pigment dispersion, coloring composition, color filter, ink for inkjet recording, and printing ink FUJIFILM CORPORATION (JP) 2013-06-25 US disclosed
US-8454710-B2 Process for producing azo compounds, pigment dispersion, coloring composition, ink for inkjet recording, coloring composition for color filter, and color filter FUJIFILM CORPORATION (JP) 2013-06-04 US disclosed
US-20130036938-A1 AZO COMPOUND, AZO PIGMENT, PIGMENT DISPERSION, COLORING COMPOSITION, COLOR FILTER, INK FOR INKJET RECORDING, AND PRINTING INK FUJIFILM CORPORATION (JP) 2013-02-14 US disclosed
US-20130000511-A1 PIGMENT COMPOSITION, INK FOR INKJET RECORDING, COLORING COMPOSITION FOR COLOR FILTER, AND COLOR FILTER FUJIFILM CORPORATION (JP) 2013-01-03 US disclosed
US-20120328984-A1 PROCESS FOR PRODUCING AZO COMPOUNDS, PIGMENT DISPERSION, COLORING COMPOSITION, INK FOR INKJET RECORDING, COLORING COMPOSITION FOR COLOR FILTER, AND COLOR FILTER FUJIFILM CORPORATION (JP) 2012-12-27 US disclosed
US-8298299-B2 Azo pigment or tautomer thereof, process for producing same, pigment dispersion, coloring composition, inkjet recording ink, coloring composition for color filter, and color filter FUJIFILM CORPORATION (JP) 2012-10-30 US disclosed
US-8298299-B2 Azo pigment or tautomer thereof, process for producing same, pigment dispersion, coloring composition, inkjet recording ink, coloring composition for color filter, and color filter FUJIFILM CORPORATION (JP) 2012-10-30 US disclosed
EP-2325264-A1 AZO COMPOUND, AZO PIGMENT, PIGMENT DISPERSION, COLOR COMPOSITION AND INK FOR INKJET RECORDING FUJIFILM Corporation (JP) 2011-05-25 EP disclosed
US-20110021764-A1 AZO PIGMENT, PIGMENT DISPERSION CONTAINING THE AZO PIGMENT, AND COLORING COMPOSITION FUJIFILM CORPORATION (JP) 2011-01-27 US disclosed
US-20110021764-A1 AZO PIGMENT, PIGMENT DISPERSION CONTAINING THE AZO PIGMENT, AND COLORING COMPOSITION FUJIFILM CORPORATION (JP) 2011-01-27 US disclosed
US-20110018946-A1 AZO COMPOUNDS, AZO PIGMENTS, AND DISPERSION, COLORING COMPOSITION AND INK FOR INKJET RECORDING CONTAINING THE AZO COMPOUNDS OR AZO PIGMENTS, INK TANK FOR INKJET RECORDING, INKJET RECORDING METHOD, AND RECORDED PRODUCTS FUJIFILM CORPORATION (JP) 2011-01-27 US disclosed
US-20110011306-A1 AZO PIGMENTS, PIGMENT DISPERSION, COLORING COMPOSITION, AND INK FOR INKJET RECORDING FUJIFILM CORPORATION (JP) 2011-01-20 US disclosed
US-20110011306-A1 AZO PIGMENTS, PIGMENT DISPERSION, COLORING COMPOSITION, AND INK FOR INKJET RECORDING FUJIFILM CORPORATION (JP) 2011-01-20 US disclosed
US-20110001777-A1 AZO COMPOUND, AZO PIGMENT, DISPERSION CONTAINING THE AZO COMPOUND OR AZO PIGMENT, COLORING COMPOSITION, INK FOR INKJET RECORDING, INK TANK FOR INKJET RECORDING, INKJET RECORDING METHOD AND RECORDED MATERIAL FUJIFILM CORPORATION (JP) 2011-01-06 US disclosed
EP-2264105-A1 AZO PIGMENT, PIGMENT DISPERSION CONTAINING THE AZO PIGMENT, AND COLORING COMPOSITION FUJIFILM Corporation (JP) 2010-12-22 EP disclosed
EP-2253672-A1 AZO COMPOUND, AZO PIGMENT, AND DISPERSION, COLORED COMPOSITION, INK-JET RECORDING INK, INK-JET RECORDING INK TANK, INK-JET RECORDING METHOD AND RECORDED MATERIAL EACH CONTAINING THE AZO COMPOUND OR THE AZO PIGMENT FUJIFILM Corporation (JP) 2010-11-24 EP disclosed
US-20100258036-A1 AZO PIGMENT, AND PIGMENT DISPERSION, COLORING COMPOSITION AND INK COMPOSITION FOR INKJET RECORDING CONTAINING THE SAME FUJIFILM CORPORATION (JP) 2010-10-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100258036-A1 AZO PIGMENT, AND PIGMENT DISPERSION, COLORING COMPOSITION AND INK COMPOSITION FOR INKJET RECORDING CONTAINING THE SAME WNT1, CYP1A1, CYP1B1 KMT2A 430/4885KDM4E 2064/4885MEN1 1329/4885
US-20130036938-A1 AZO COMPOUND, AZO PIGMENT, PIGMENT DISPERSION, COLORING COMPOSITION, COLOR FILTER, INK FOR INKJET RECORDING, AND PRINTING INK RB1, CRY1, TYR KMT2A 203/4885KDM4E 2692/4885MEN1 888/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.