SCHEMBL8247100

SCHEMBL8247100

C=CCOC(=O)c1ccc2c(c1C)CC[C@@H]2NC(=O)c1cc(C(=O)NC(C)C2CC=C(C#N)S2)nc2ncnn12

nearest known ligand 0.37

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADAMTS4 O75173 2/20 0.37
MMP3 P08254 2/20 0.37
MMP13 P45452 2/20 0.37
MMP8 P22894 1/20 0.35
MMP12 P39900 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8246538 0.89 ADAMTS4 (0.45) ADAMTS4MMP3MMP13MMP8MMP12
SCHEMBL8254358 0.88 ADAMTS4 (0.40) ADAMTS4MMP3MMP13MMP8MMP12
SCHEMBL10165457 0.84 ADAMTS4 (0.36) ADAMTS4MMP3MMP13MMP8MMP12
SCHEMBL8246226 0.82 ADAMTS4 (0.45) ADAMTS4MMP3MMP13MMP8MMP12
SCHEMBL8246504 0.82 ADAMTS4 (0.41) ADAMTS4MMP3MMP13MMP8MMP12
SCHEMBL8255480 0.82 ADAMTS4 (0.41) ADAMTS4MMP3MMP13MMP8MMP12
SCHEMBL8253969 0.81 ADAMTS4 (0.44) ADAMTS4MMP3MMP13MMP8MMP12
SCHEMBL10165450 0.81 ADAMTS4 (0.48) ADAMTS4MMP3MMP13MMP8MMP12
SCHEMBL10165436 0.81 ADAMTS4 (0.42) ADAMTS4MMP3MMP13MMP8MMP12
SCHEMBL10165452 0.80 MMP13 (0.47) ADAMTS4MMP3MMP13MMP8MMP12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006128184-A2 PYRIMIDINE OR TRIAZINE FUSED BICYCLIC METALLOPROTEASE INHIBITORS ALANTOS-PHARMACEUTICALS, INC. (US) 2006-11-30 WO disclosed