SCHEMBL8247227

SCHEMBL8247227

Cc1c(C(=O)O)ccc2c1CC[C@@H]2NC(=O)c1cc(C(=O)NCc2ccnc(N)c2)nc2c(F)cnn12

nearest known ligand 0.77

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ADAMTS4 O75173 2/20 0.77
MMP3 P08254 2/20 0.77
MMP13 P45452 2/20 0.77
MMP8 P22894 1/20 0.56
MMP12 P39900 1/20 0.56
KLKB1 P03952 6/20 0.37
NTRK1 P04629 7/20 0.35
DHODH Q02127 2/20 0.33
SLC8A1 P32418 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8256338 0.91 MMP13 (0.82) ADAMTS4MMP3MMP13MMP8MMP12
SCHEMBL8256275 0.90 MMP13 (0.86) ADAMTS4MMP3MMP13MMP8MMP12
SCHEMBL10166038 0.90 MMP13 (0.74) ADAMTS4MMP3MMP13MMP8MMP12
SCHEMBL8222933 0.90 MMP13 (0.80) ADAMTS4MMP3MMP13MMP8MMP12
SCHEMBL10166080 0.89 MMP13 (0.82) ADAMTS4MMP3MMP13MMP8MMP12
SCHEMBL8255754 0.89 MMP13 (0.80) ADAMTS4MMP3MMP13MMP8MMP12
SCHEMBL8252163 0.89 ADAMTS4 (0.62) ADAMTS4MMP3MMP13MMP8MMP12
SCHEMBL8253462 0.89 MMP13 (0.81) ADAMTS4MMP3MMP13MMP8MMP12
SCHEMBL10167263 0.89 ADAMTS4 (0.73) ADAMTS4MMP3MMP13MMP8MMP12
SCHEMBL8246527 0.88 MMP13 (0.76) ADAMTS4MMP3MMP13MMP8MMP12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006128184-A2 PYRIMIDINE OR TRIAZINE FUSED BICYCLIC METALLOPROTEASE INHIBITORS ALANTOS-PHARMACEUTICALS, INC. (US) 2006-11-30 WO disclosed