SCHEMBL8247779

SCHEMBL8247779

NC12CCC(CNC(=O)c3cc(C(=O)NCc4ccc(F)c(Cl)c4)nc4ncnn34)(CC1)CC2

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 3/20 0.39
MAPK1 P28482 9/20 0.39
PDE2A O00408 3/20 0.37
RPS6KA1 Q15418 1/20 0.37
DGAT1 O75907 1/20 0.36
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
BCDIN3D Q7Z5W3 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10165622 0.94 MMP13 (0.39) MMP13MAPK1PDE2ARPS6KA1DGAT1
SCHEMBL8225272 0.93 MMP13 (0.40) MMP13MAPK1PDE2ARPS6KA1DGAT1
SCHEMBL10162252 0.92 MMP13 (0.40) MMP13MAPK1PDE2ARPS6KA1DGAT1
SCHEMBL10165624 0.92 MMP13 (0.39) MMP13MAPK1PDE2ARPS6KA1DGAT1
SCHEMBL8256775 0.92 MMP13 (0.39) MMP13MAPK1PDE2ARPS6KA1DGAT1
SCHEMBL10162208 0.92 MMP13 (0.41) MMP13MAPK1PDE2ARPS6KA1DGAT1
SCHEMBL10209873 0.91 MMP13 (0.40) MMP13MAPK1PDE2ARPS6KA1DGAT1
SCHEMBL8255580 0.91 MMP13 (0.39) MMP13MAPK1PDE2ARPS6KA1DGAT1
SCHEMBL10165620 0.90 MMP13 (0.38) MMP13MAPK1PDE2ARPS6KA1DGAT1
SCHEMBL10165797 0.88 MMP13 (0.46) MMP13MAPK1PDE2ARPS6KA1DGAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006128184-A2 PYRIMIDINE OR TRIAZINE FUSED BICYCLIC METALLOPROTEASE INHIBITORS ALANTOS-PHARMACEUTICALS, INC. (US) 2006-11-30 WO disclosed