SCHEMBL8248263

SCHEMBL8248263

CC1(C)CCc2nc(-n3cnc(-c4cccc(N)c4)c3)ccc2C1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.40
ALDH1A1 P00352 2/20 0.33
POLB P06746 1/20 0.33
GFER P55789 1/20 0.33
BRD4 O60885 1/20 0.32
AKT1 P31749 2/20 0.32
AKT2 P31751 2/20 0.32
AKT3 Q9Y243 2/20 0.32
ATR Q13535 1/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
TSHR P16473 1/20 0.32
RECQL P46063 1/20 0.32
MAPT P10636 2/20 0.31
LMNA P02545 2/20 0.31
TP53 P04637 1/20 0.31
TDP2 O95551 1/20 0.31
RAD52 P43351 1/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4684250 0.94 GRM5 (0.40) GRM5ALDH1A1POLBGFERBRD4
SCHEMBL4686098 0.85 GRM5 (0.44) GRM5ALDH1A1BRD4CYP11B2CHEK1
SCHEMBL4683088 0.85 GRM5 (0.37) GRM5GSK3B
SCHEMBL6103021 0.83 GRM5 (0.40) GRM5ALDH1A1POLBGFERBRD4
SCHEMBL4679372 0.82 GRM5 (0.40) GRM5ALDH1A1TSHRMAPTLMNA
SCHEMBL4686152 0.80 GRM5 (0.36) GRM5CYP11B2
SCHEMBL4686025 0.79 GRM5 (0.40) GRM5AKT1AKT2CYP11B2
SCHEMBL4736631 0.77 GRM5 (0.34) GRM5
SCHEMBL4686336 0.76 CYP11B2 (0.40) GRM5CYP11B2
SCHEMBL4684400 0.74 CYP11B2 (0.40) GRM5CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007023245-A1 TETRAHYDROQUINOLINONES AND THEIR USE AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS MERZ PHARMA GMBH & CO. KGAA (DE) 2007-03-01 WO disclosed