SCHEMBL8249796

SCHEMBL8249796

CC(C)(C)CCn1c(=O)c(C(=O)NCC(=O)O)c(O)c2cc(F)ccc21

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 15/20 0.58
EGLN3 Q9H6Z9 2/20 0.56
EGLN1 Q9GZT9 3/20 0.53
L3MBTL1 Q9Y468 1/20 0.50
EGLN2 Q96KS0 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8245606 0.94 HIF1A (0.56) HIF1AEGLN3EGLN1L3MBTL1EGLN2
SCHEMBL8248316 0.93 HIF1A (0.55) HIF1AEGLN3EGLN1L3MBTL1EGLN2
SCHEMBL8248071 0.86 HIF1A (0.56) HIF1AEGLN3EGLN1L3MBTL1
SCHEMBL8243641 0.85 HIF1A (0.67) HIF1AEGLN3EGLN1EGLN2
SCHEMBL2382549 0.84 HIF1A (0.72) HIF1AEGLN1
SCHEMBL8237955 0.84 EGLN1 (0.64) HIF1AEGLN3EGLN1L3MBTL1
SCHEMBL8247183 0.83 HIF1A (0.62) HIF1AEGLN3EGLN1EGLN2
SCHEMBL8245604 0.82 HIF1A (0.61) HIF1AEGLN3EGLN1EGLN2
SCHEMBL8247330 0.82 EGLN1 (0.65) HIF1AEGLN3EGLN1L3MBTL1EGLN2
SCHEMBL8244124 0.82 EGLN1 (0.59) HIF1AEGLN3EGLN1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007038571-A2 PROLYL HYDROXYLASE ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2007-04-05 WO disclosed