SCHEMBL8245604

SCHEMBL8245604

O=C(O)CNC(=O)c1c(O)c2cc(F)ccc2n(CCC2CCCCC2)c1=O

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 11/20 0.61
EGLN3 Q9H6Z9 3/20 0.51
EGLN1 Q9GZT9 6/20 0.47
EGLN2 Q96KS0 2/20 0.47
BBOX1 O75936 1/20 0.45
ASPH Q12797 1/20 0.45
KDM8 Q8N371 1/20 0.45
NR1I2 O75469 1/20 0.44
CYP2C9 P11712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8247183 0.99 HIF1A (0.62) HIF1AEGLN3EGLN1EGLN2BBOX1
SCHEMBL8243641 0.95 HIF1A (0.67) HIF1AEGLN3EGLN1EGLN2BBOX1
SCHEMBL8237984 0.86 HIF1A (0.68) HIF1AEGLN1BBOX1ASPHKDM8
SCHEMBL8249796 0.82 HIF1A (0.58) HIF1AEGLN3EGLN1EGLN2
SCHEMBL5308270 0.81 HIF1A (0.74) HIF1AEGLN1BBOX1ASPHKDM8
SCHEMBL8245606 0.81 HIF1A (0.56) HIF1AEGLN3EGLN1EGLN2
SCHEMBL8248071 0.81 HIF1A (0.56) HIF1AEGLN3EGLN1
SCHEMBL8237955 0.81 EGLN1 (0.64) HIF1AEGLN3EGLN1
SCHEMBL5330885 0.80 ALDH1A1 (0.56) HIF1ANR1I2CYP2C9
SCHEMBL8248316 0.80 HIF1A (0.55) HIF1AEGLN3EGLN1EGLN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007038571-A2 PROLYL HYDROXYLASE ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2007-04-05 WO disclosed