SCHEMBL8250133

SCHEMBL8250133

C=CC1C[C@]1(NC(=O)[C@@H]1C[C@@H](Oc2cc(-c3nc(C(C)C)cs3)nc3cc(OC)ccc23)CN1)C(=O)OCC

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSB P07858 1/20 0.36
PPP3CB P16298 1/20 0.36
CTSS P25774 1/20 0.34
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8250198 1.00 CTSB (0.36) CTSBPPP3CBCTSSCYP3A4
SCHEMBL3277398 1.00 CTSB (0.36) CTSBPPP3CBCTSSCYP3A4
SCHEMBL12383127 0.91 CTSS (0.35) CTSS
SCHEMBL11888410 0.91 CTSS (0.35) CTSS
SCHEMBL10156683 0.90 CTSS (0.42) CTSBPPP3CBCTSS
SCHEMBL2449092 0.89 CTSB (0.35) CTSBPPP3CBCTSSCYP3A4
SCHEMBL11887180 0.89 CTSB (0.35) CTSBPPP3CBCTSSCYP3A4
SCHEMBL13385448 0.88 CTSS (0.35) CTSS
SCHEMBL2212114 0.88 CTSB (0.41) CTSBPPP3CBCTSS
SCHEMBL8248937 0.88 CTSB (0.41) CTSBPPP3CBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007017144-A2 MACROCYLIC INHIBITORS OF HEPATITIS C VIRUS MEDIVIR AB (SE) 2007-02-15 WO disclosed