SCHEMBL8250583

SCHEMBL8250583

CCCCNC(=O)n1ccc2c(Cc3c[nH]c4ncc(C5C=NN(C)C5)cc34)cccc21

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ASAH1 Q13510 2/20 0.33
CYP3A4 P08684 1/20 0.31
MAP4K1 Q92918 1/20 0.31
JAK2 O60674 1/20 0.30
JAK1 P23458 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL858744 0.81 ALK (0.43) CYP3A4MAP4K1
SCHEMBL8249506 0.81 MTNR1B (0.48) ASAH1CYP3A4
SCHEMBL8242206 0.79 AXL (0.41) ASAH1CYP3A4MAP4K1
SCHEMBL8249503 0.78 CYP3A4 (0.40) ASAH1CYP3A4MAP4K1
SCHEMBL413921 0.78 PDPK1 (0.42) CYP3A4MAP4K1
SCHEMBL14620858 0.77 ASAH1 (0.34) ASAH1CYP3A4MAP4K1
SCHEMBL17170056 0.76 MTNR1A (0.39) ASAH1CYP3A4MAP4K1
SCHEMBL859405 0.72 MAPT (0.32) ASAH1CYP3A4MAP4K1
SCHEMBL858516 0.72 SNCA (0.39) CYP3A4MAP4K1JAK2
SCHEMBL10257418 0.71 MTNR1B (0.43) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007002325-A1 PYRROLO[2,3-B] PYRIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS PLEXXIKON, INC. (US) 2007-01-04 WO disclosed