SCHEMBL8251165

SCHEMBL8251165

O=C(O)c1cccc(S(=O)(=O)Nc2cccc(Cl)c2)c1

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PFKFB3 Q16875 1/20 0.67
MEN1 O00255 4/20 0.66
KMT2A Q03164 4/20 0.66
TSHR P16473 2/20 0.66
ALDH1A1 P00352 1/20 0.66
PGR P06401 2/20 0.66
AKR1C3 P42330 2/20 0.65
POLB P06746 2/20 0.63
KDM4E B2RXH2 1/20 0.63
PTK2B Q14289 1/20 0.63
THRB P10828 1/20 0.60
MAPT P10636 3/20 0.60
HSD17B10 Q99714 1/20 0.60
LMNA P02545 1/20 0.59
PTBP1 P26599 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29875309 0.94 PFKFB3 (0.71) PFKFB3MEN1KMT2ATSHRALDH1A1
SCHEMBL2831061 0.94 PFKFB3 (0.71) PFKFB3MEN1KMT2ATSHRALDH1A1
SCHEMBL29369447 0.94 PFKFB3 (0.71) PFKFB3MEN1KMT2ATSHRALDH1A1
SCHEMBL7365696 0.90 KDM4E (0.64) PFKFB3MEN1KMT2ATSHRPGR
SCHEMBL7366821 0.87 AKR1C3 (0.67) PFKFB3MEN1KMT2ATSHRPGR
SCHEMBL664321 0.87 KMT2A (0.75) MEN1KMT2ATSHRALDH1A1PGR
SCHEMBL30702318 0.86 PFKFB3 (0.76) PFKFB3MEN1KMT2ATSHRAKR1C3
SCHEMBL4063367 0.86 PFKFB3 (0.76) PFKFB3MEN1KMT2ATSHRAKR1C3
SCHEMBL30702319 0.86 PFKFB3 (0.76) PFKFB3MEN1KMT2ATSHRAKR1C3
SCHEMBL8241750 0.85 TCF4 (0.64) PFKFB3MEN1KMT2ATSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504431-B2 Sulfonyl amide inhibitors of calcium channel function BRISTOL-MYERS SQUIBB COMPANY (US) 2009-03-17 US disclosed
US-7504431-B2 Sulfonyl amide inhibitors of calcium channel function BRISTOL-MYERS SQUIBB COMPANY (US) 2009-03-17 US disclosed
US-20050245535-A1 Sulfonyl amide inhibitors of calcium channel function BRISTOL- MYERS SQUIBB COMPANY 2005-11-03 US disclosed
US-20050245535-A1 Sulfonyl amide inhibitors of calcium channel function BRISTOL- MYERS SQUIBB COMPANY 2005-11-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050245535-A1 Sulfonyl amide inhibitors of calcium channel function CACNA1F, CACNA1A, CACNA1D PFKFB3 2451/4885MEN1 2007/4885KMT2A 3232/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.