SCHEMBL8255902

SCHEMBL8255902

Cc1cc(CN)ccc1C(=O)CC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
NCOR2 Q9Y618 1/20 0.39
PLG P00747 3/20 0.38
KLK1 P06870 3/20 0.38
KLK6 Q92876 3/20 0.38
LOXL2 Q9Y4K0 2/20 0.38
GRM2 Q14416 1/20 0.36
S1PR1 P21453 1/20 0.36
KLKB1 P03952 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL507659 0.83 CSNK2A1 (0.40) NR1H4LOXL2KLKB1
SCHEMBL507089 0.83 LOXL2 (0.43) NR1H4LOXL2
SCHEMBL12933288 0.80 HSD11B1 (0.50)
SCHEMBL1146167 0.78 NR1H4 (0.50) NR1H4HDAC3HDAC6NCOR2PLG
SCHEMBL6224042 0.78 MKNK1 (0.44) HDAC3HDAC6NCOR2PLGKLK1
SCHEMBL506919 0.78 HDAC3 (0.53) HDAC3HDAC6NCOR2LOXL2
SCHEMBL8246361 0.76 LOXL2 (0.44) NR1H4PLGKLK1KLK6LOXL2
Hydrochloric Acid SCHEMBL479729 0.76 NR1H4 (0.49) NR1H4PLGKLK1KLK6LOXL2
SCHEMBL3174714 0.73 LOXL2 (0.61) HDAC3HDAC6NCOR2PLGKLK1
Hydrochloric Acid SCHEMBL12499723 0.72 LOXL2 (0.59) PLGKLK1KLK6LOXL2KLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006128184-A2 PYRIMIDINE OR TRIAZINE FUSED BICYCLIC METALLOPROTEASE INHIBITORS ALANTOS-PHARMACEUTICALS, INC. (US) 2006-11-30 WO disclosed