SCHEMBL8258749

SCHEMBL8258749

COc1ccc2c(c1)CC(I)N2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.44
PDE3A Q14432 2/20 0.44
DRD2 P14416 1/20 0.41
DRD3 P35462 1/20 0.41
EGFR P00533 1/20 0.41
PDGFRA P16234 1/20 0.41
KDR P35968 1/20 0.41
CHRNB2 P17787 1/20 0.40
CHRNB4 P30926 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA7 P36544 1/20 0.40
CHRNA4 P43681 1/20 0.40
ALDH1A1 P00352 1/20 0.40
SNCA P37840 1/20 0.40
HTR2C P28335 1/20 0.39
GAA P10253 1/20 0.39
BCL2 P10415 1/20 0.39
ACHE P22303 1/20 0.38
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13937919 0.88 HTR5A (0.44) PDE3BPDE3ADRD2DRD3CHRNB2
SCHEMBL7309997 0.82 PDE3B (0.41) PDE3BPDE3ADRD2DRD3EGFR
SCHEMBL11087883 0.81 PDE3B (0.45) PDE3BPDE3ADRD2DRD3EGFR
Hydrochloric Acid SCHEMBL7313862 0.81 PDE3B (0.40) PDE3BPDE3AEGFRPDGFRAKDR
SCHEMBL7297564 0.76 PDE3B (0.41) PDE3BPDE3ADRD2DRD3EGFR
SCHEMBL8399480 0.76 PDE3B (0.44) PDE3BPDE3ADRD2DRD3EGFR
SCHEMBL7297572 0.76 PDE3B (0.41) PDE3BPDE3ADRD2DRD3EGFR
SCHEMBL7037302 0.74 GAA (0.55) PDE3BPDE3AALDH1A1GAAACHE
SCHEMBL11699617 0.74 SLC6A2 (0.44) GAAMAOBCYP19A1
SCHEMBL4365304 0.74 GAA (0.55) PDE3BPDE3AALDH1A1GAAACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006102760-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2006-10-05 WO disclosed