SCHEMBL8259359

SCHEMBL8259359

O=CC(Cc1ccccc1)NC(=O)C(Cc1ccccc1)NC(=O)OCc1ccccc1

nearest known ligand 0.74

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSL P07711 7/20 0.70
CTSB P07858 5/20 0.70
CTSS P25774 3/20 0.69
TACR1 P25103 2/20 0.64
CTSK P43235 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23234615 1.00 CTSL (0.70) CTSLCTSBCTSSTACR1CTSK
SCHEMBL4409560 1.00 CTSL (0.70) CTSLCTSBCTSSTACR1CTSK
SCHEMBL14513407 0.95 CTSL (0.65) CTSLCTSBCTSSTACR1
SCHEMBL7028199 0.95 CTSL (0.65) CTSLCTSBCTSSTACR1
SCHEMBL7028202 0.95 CTSL (0.65) CTSLCTSBCTSSTACR1
SCHEMBL2245863 0.90 CTSL (0.68) CTSLCTSBCTSS
SCHEMBL7027265 0.90 CTSL (0.75) CTSLCTSBCTSS
SCHEMBL7027268 0.90 CTSL (0.75) CTSLCTSBCTSS
SCHEMBL8261584 0.90 CTSL (0.68) CTSLCTSBCTSS
SCHEMBL7027261 0.90 CTSL (0.75) CTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7589066-B2 Such as N-carbobenzyloxy-phenylalanyl-phenylalanylal; for treating cancer, inflammation, and/or autoimmune diseases; suppresses endogenous antigenic peptide generation THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2009-09-15 US disclosed
US-7589066-B2 Such as N-carbobenzyloxy-phenylalanyl-phenylalanylal; for treating cancer, inflammation, and/or autoimmune diseases; suppresses endogenous antigenic peptide generation THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2009-09-15 US disclosed
WO-2006099261-A2 POTENT AND SPECIFIC IMMUNOPROTEASOME INHIBITORS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2006-09-21 WO disclosed