SCHEMBL8263144

SCHEMBL8263144

COCCCOc1cc(CN(C[C@@H]2CCNC2)C(C)C)ccc1OC

nearest known ligand 0.65

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
REN P00797 19/20 0.65
KCNH2 Q12809 3/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
SLC6A2 P23975 1/20 0.45
SLC6A4 P31645 1/20 0.45
CYP2C19 P33261 1/20 0.45
SLC6A3 Q01959 1/20 0.45
HTR1A P08908 2/20 0.44
ADRA1D P25100 2/20 0.44
HTR2A P28223 2/20 0.44
ADRA1A P35348 2/20 0.44
ADRA1B P35368 2/20 0.44
HTR2B P41595 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13177323 0.81 REN (0.67) RENKCNH2SLC6A2SLC6A4SLC6A3
SCHEMBL13177128 0.79 REN (1.00) RENKCNH2CYP3A4HTR1AADRA1D
SCHEMBL2934673 0.79 REN (1.00) RENKCNH2CYP3A4HTR1AADRA1D
SCHEMBL2929532 0.78 REN (0.67) RENKCNH2CYP3A4HTR1AADRA1D
SCHEMBL8262709 0.78 REN (0.67) RENKCNH2CYP3A4HTR1AADRA1D
SCHEMBL8262513 0.78 REN (0.67) RENKCNH2CYP3A4HTR1AADRA1D
SCHEMBL1911550 0.70 REN (1.00) RENKCNH2
SCHEMBL4323431 0.70 SLC6A2 (0.57) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL3487650 0.69 REN (0.56) RENKCNH2SLC6A2SLC6A4HTR1A
SCHEMBL8263200 0.69 REN (0.54) RENKCNH2HTR1AADRA1DHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006066896-A2 PYRROLIDINE DERIVATIVES FOR THE TREATMENT OF A DISEASE DEPENDING ON THE ACTIVITY OF RENIN NOVARTIS AG (CH) 2006-06-29 WO disclosed