Mtic

Mtic

SCHEMBL826375

C/N=N/Nc1[nH]cnc1C(N)=O

nearest known ligand 0.36

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Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GDA Q9Y2T3 1/20 0.36
LMNA P02545 2/20 0.35
TSHR P16473 2/20 0.35
PAX8 Q06710 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MMP9 P14780 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
GAA P10253 3/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
XDH P47989 1/20 0.31
MAPT P10636 1/20 0.31
PARP1 P09874 1/20 0.31
CYP2C19 P33261 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Mtic SCHEMBL22757309 1.00 GDA (0.36) GDALMNATSHRPAX8KDM4E
SCHEMBL28386283 0.75 GDA (0.37) GDALMNATSHRPAX8KDM4E
SCHEMBL15131350 0.75 GDA (0.39) GDALMNATSHRPAX8KDM4E
SCHEMBL18737907 0.74 PAX8 (0.38) GDALMNATSHRPAX8KDM4E
SCHEMBL13348562 0.74 GDA (0.41) GDALMNATSHRPAX8KDM4E
SCHEMBL14034284 0.74 GDA (0.41) GDALMNATSHRPAX8KDM4E
SCHEMBL12259351 0.73 MAPK1 (0.40) GDAPAX8SMN1; SMN2
SCHEMBL28543470 0.73 GDA (0.40) GDAKDM4EALDH1A1SMN1; SMN2GAA
SCHEMBL4210787 0.71 GDA (0.39) GDALMNATSHRPAX8KDM4E
SCHEMBL1059195 0.71 GDA (0.39) GDALMNATSHRPAX8KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8258119-B2 Anti-cancer drugs and uses relating thereto for metastatic malignant melanoma and other cancers Kasina Laila Innova Pharmaceuticals (IN) 2012-09-04 US disclosed
US-8258119-B2 Anti-cancer drugs and uses relating thereto for metastatic malignant melanoma and other cancers Kasina Laila Innova Pharmaceuticals (IN) 2012-09-04 US disclosed
US-8143237-B2 Anti-cancer drugs, and uses relating for malignant melanoma and other cancers KASINA LAILA INNOVA PHARMACEUTICALS PRIVATE LIMITED (US) 2012-03-27 US disclosed
US-8143237-B2 Anti-cancer drugs, and uses relating for malignant melanoma and other cancers KASINA LAILA INNOVA PHARMACEUTICALS PRIVATE LIMITED (US) 2012-03-27 US disclosed
US-20100272678-A1 ANTI-CANCER DRUGS, AND USES RELATING FOR MALIGNANT MELANOMA AND OTHER CANCERS KASINA LAILA INNOVA PHARMACEUTICALS PRIVATE LIMITE (IN) 2010-10-28 US disclosed
US-20100272678-A1 ANTI-CANCER DRUGS, AND USES RELATING FOR MALIGNANT MELANOMA AND OTHER CANCERS KASINA LAILA INNOVA PHARMACEUTICALS PRIVATE LIMITE (IN) 2010-10-28 US disclosed
US-20100068178-A1 ANTI-CANCER DRUGS AND USES RELATING THERETO FOR METASTATIC MALIGNANT MELANOMA AND OTHER CANCERS LAILA NUTRACEUTICALS (IN) 2010-03-18 US disclosed
US-20100068178-A1 ANTI-CANCER DRUGS AND USES RELATING THERETO FOR METASTATIC MALIGNANT MELANOMA AND OTHER CANCERS LAILA NUTRACEUTICALS (IN) 2010-03-18 US disclosed
US-7572798-B2 Prevent Dna damage; antitumor, anticancer agents; blocking epidermal growth factor receptor MCGILL UNIVERSITY (CA) 2009-08-11 US disclosed
US-7572798-B2 Prevent Dna damage; antitumor, anticancer agents; blocking epidermal growth factor receptor MCGILL UNIVERSITY (CA) 2009-08-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100272678-A1 ANTI-CANCER DRUGS, AND USES RELATING FOR MALIGNANT MELANOMA AND OTHER CANCERS BRAF, TPD52L2, SALL4 GDA 4395/4885LMNA 3063/4885TSHR 74/4885
US-20100068178-A1 ANTI-CANCER DRUGS AND USES RELATING THERETO FOR METASTATIC MALIGNANT MELANOMA AND OTHER CANCERS BRAF, NRAS, TP53 GDA 1130/4885LMNA 1600/4885TSHR 2319/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.