SCHEMBL8265997

SCHEMBL8265997

O=Cc1cc(Sc2cccc(N[S+]([O-])c3ccccc3)c2)ccc1[N+](=O)[O-]

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT5 Q9NXA8 2/20 0.37
MEN1 O00255 6/20 0.34
KMT2A Q03164 6/20 0.34
MAPT P10636 5/20 0.34
ALDH1A1 P00352 4/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
ERN1 O75460 3/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
KDM4E B2RXH2 2/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
PDE7A Q13946 2/20 0.33
PDE7B Q9NP56 1/20 0.33
TDP1 Q9NUW8 2/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8266752 0.80 MEN1 (0.35) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL8271839 0.79 ALDH1A1 (0.40) SIRT5MEN1KMT2AMAPTALDH1A1
SCHEMBL2931113 0.78 GAA (0.51) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL8272311 0.74 MEN1 (0.33) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL10478056 0.70 PDE7A (0.47) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL2932238 0.67 FFAR4 (0.49) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL9668230 0.66 ALDH1A1 (0.47) MEN1KMT2AMAPTALDH1A1ERN1
SCHEMBL8272607 0.65 SLC6A4 (0.38) KMT2AALDH1A1
SCHEMBL10477862 0.64 MEN1 (0.44) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL8272305 0.63 ALDH1A1 (0.38) MEN1KMT2AMAPTALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006024932-A1 2-AMINO-QUINAZOLINE DERIVATIVES USEFUL AS INHIBITORS OF B-SECRETASE (BACE) JANSSEN PHARMACEUTICA, N.V. (US) 2006-03-09 WO disclosed
WO-2006017844-A1 NOVEL 2-AMINO-QUINAZOLINE DERIVATIVES USEFUL AS INHIBITORS OF β-SECRETASE (BACE) JANSSEN PHARMACEUTICA, N.V. (BE) 2006-02-16 WO disclosed
WO-2006017836-A2 2-AMINO-QUINAZOLINE DERIVATIVES USEFUL AS INHIBITORS OF BETA-SECRETASE (BACE) JANSSEN PHARMACEUTICA, N.V. (BE) 2006-02-16 WO disclosed