SCHEMBL8266752

SCHEMBL8266752

COC(OC)c1cc(Sc2cccc(N[S+]([O-])c3ccccc3)c2)ccc1[N+](=O)[O-]

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.35
KMT2A Q03164 5/20 0.35
MAPT P10636 5/20 0.35
TDP1 Q9NUW8 2/20 0.35
HTT P42858 1/20 0.34
ALDH1A1 P00352 6/20 0.34
KDM4E B2RXH2 1/20 0.32
ABCC9 O60706 1/20 0.32
ABCC8 Q09428 1/20 0.32
KCNJ11 Q14654 1/20 0.32
KCNJ8 Q15842 1/20 0.32
AKR1C4 P17516 1/20 0.32
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32
AKR1C1 Q04828 1/20 0.32
CYP3A4 P08684 1/20 0.32
TSHR P16473 1/20 0.32
PDE7A Q13946 2/20 0.31
PDE7B Q9NP56 1/20 0.31
NPC1 O15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8272305 0.84 ALDH1A1 (0.38) MEN1KMT2AMAPTTDP1HTT
SCHEMBL2928164 0.81 HPGD (0.50) MEN1KMT2AMAPTHTTALDH1A1
SCHEMBL8265997 0.80 SIRT5 (0.37) MEN1KMT2AMAPTTDP1HTT
SCHEMBL2932823 0.77 PDE7A (0.49) MEN1KMT2AMAPTTDP1ALDH1A1
SCHEMBL8271839 0.77 ALDH1A1 (0.40) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL8272056 0.74 ALDH1A1 (0.39) MEN1KMT2AMAPTTDP1HTT
SCHEMBL8267130 0.70 FFAR1 (0.38) MEN1KMT2AMAPTHTTALDH1A1
SCHEMBL3362982 0.65 ALDH1A1 (0.43) MEN1KMT2AMAPTTDP1HTT
SCHEMBL15481223 0.65 HTT (0.44) MEN1KMT2AMAPTTDP1HTT
SCHEMBL2904377 0.65 ALDH1A1 (0.56) MEN1KMT2AMAPTTDP1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006017844-A1 NOVEL 2-AMINO-QUINAZOLINE DERIVATIVES USEFUL AS INHIBITORS OF β-SECRETASE (BACE) JANSSEN PHARMACEUTICA, N.V. (BE) 2006-02-16 WO disclosed
WO-2006017836-A2 2-AMINO-QUINAZOLINE DERIVATIVES USEFUL AS INHIBITORS OF BETA-SECRETASE (BACE) JANSSEN PHARMACEUTICA, N.V. (BE) 2006-02-16 WO disclosed