SCHEMBL8267274

SCHEMBL8267274

CN1OC(C)(c2cccc(-c3cccc(N)c3)c2)NC1=N

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.37
BACE1 P56817 6/20 0.33
MAP4K4 O95819 5/20 0.33
BRD4 O60885 1/20 0.32
MEN1 O00255 1/20 0.32
PSIP1 O75475 1/20 0.32
AXL P30530 1/20 0.32
MKNK1 Q9BUB5 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32
PRKCA P17252 1/20 0.32
GSK3B P49841 1/20 0.32
NPY5R Q15761 1/20 0.32
PDPK1 O15530 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2171684 0.84 BACE1 (0.43) BACE1
SCHEMBL2173280 0.84 PGR (0.40) BACE1NPY5R
SCHEMBL8412303 0.84 HSD17B2 (0.38)
SCHEMBL2175983 0.83 BACE1 (0.38) BACE1
SCHEMBL2175281 0.82 BACE1 (0.45) BACE1BRD4
SCHEMBL14643302 0.81
SCHEMBL2171800 0.81 BACE1 (0.47) BACE1MEN1PSIP1AXLMKNK1
SCHEMBL13663905 0.80 BACE1 (0.33) BACE1GSK3B
SCHEMBL13663904 0.80 HTR7 (0.38) BACE1
SCHEMBL2174928 0.79 PGR (0.38) BACE1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006065277-A2 HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS SCHERING CORPORATION (US) 2006-06-22 WO disclosed