SCHEMBL8268366

SCHEMBL8268366

CCOC(=O)CCCNc1nc(-c2ccc(-c3cccc(C(F)(F)F)c3)cc2)nc2ccccc12

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 3/20 0.76
MAPT P10636 4/20 0.53
KDM4E B2RXH2 4/20 0.53
GBA1 P04062 3/20 0.53
MEN1 O00255 3/20 0.53
KMT2A Q03164 3/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
ALDH1A1 P00352 1/20 0.53
TP53 P04637 1/20 0.53
TOP2A P11388 1/20 0.52
HPGD P15428 1/20 0.52
RECQL P46063 2/20 0.51
ACP1 P24666 1/20 0.51
ABCG2 Q9UNQ0 1/20 0.49
SIRT5 Q9NXA8 1/20 0.49
POLB P06746 2/20 0.48
PKM P14618 2/20 0.48
LMNA P02545 1/20 0.48
ELANE P08246 1/20 0.48
CYP1A2 P05177 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8270099 0.95 PDE5A (0.67) PDE5AMAPTKDM4EGBA1MEN1
SCHEMBL8268899 0.91 PDE5A (0.61) PDE5AMAPTKDM4EGBA1MEN1
SCHEMBL8268384 0.88 SIRT5 (0.61) PDE5AMAPTKDM4EGBA1MEN1
SCHEMBL1085482 0.87 PDE5A (1.00) PDE5AMAPTKDM4EGBA1MEN1
SCHEMBL8268895 0.85 PDE5A (0.54) PDE5AMAPTKDM4EGBA1MEN1
SCHEMBL8270100 0.84 ACP1 (0.55) PDE5ATOP2AACP1ELANE
SCHEMBL8269549 0.82 PDE5A (0.86) PDE5AMAPTKDM4EGBA1MEN1
SCHEMBL8269560 0.79 PDE10A (0.58) TOP2AACP1
SCHEMBL8268382 0.79 ABCG2 (0.57) PDE5AACP1ABCG2SIRT5CYP1A2
SCHEMBL8269905 0.79 SIRT5 (0.47) PDE5AABCG2SIRT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006034512-A2 PHENYL-SUBSTITUTED QUINOLINE AND QUINAZOLINE COMPOUNDS FOR THE TREATMENT OF DIABETES BAYER PHARMACEUTICALS CORPORATION (US) 2006-03-30 WO disclosed