SCHEMBL8268384

SCHEMBL8268384

O=C(O)CCCNc1nc(-c2ccc(-c3cccc(C(F)(F)F)c3)cc2)nc2ccccc12

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT5 Q9NXA8 2/20 0.61
PDE5A O76074 3/20 0.56
ABCG2 Q9UNQ0 3/20 0.55
ACP1 P24666 1/20 0.52
KMT2A Q03164 4/20 0.52
MEN1 O00255 3/20 0.50
MAPK1 P28482 2/20 0.50
RECQL P46063 2/20 0.49
MAPT P10636 2/20 0.49
KDM4E B2RXH2 2/20 0.49
GBA1 P04062 1/20 0.49
TLR9 Q9NR96 1/20 0.49
LATS1 O95835 1/20 0.48
LMNA P02545 1/20 0.48
POLB P06746 1/20 0.48
PKM P14618 1/20 0.48
ALDH1A1 P00352 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8269905 0.90 SIRT5 (0.47) SIRT5PDE5AABCG2LATS1
SCHEMBL8268366 0.88 PDE5A (0.76) SIRT5PDE5AABCG2ACP1KMT2A
SCHEMBL8270099 0.84 PDE5A (0.67) SIRT5PDE5AABCG2ACP1KMT2A
SCHEMBL8268382 0.84 ABCG2 (0.57) SIRT5PDE5AABCG2ACP1MAPK1
SCHEMBL8271003 0.82 PDE10A (0.62) ACP1
SCHEMBL5530299 0.80 SIRT5 (0.70) SIRT5PDE5AACP1KMT2AMEN1
SCHEMBL8268899 0.79 PDE5A (0.61) PDE5AABCG2KMT2AMEN1MAPT
SCHEMBL4867588 0.78 PDE5A (0.71) SIRT5PDE5AABCG2ACP1KMT2A
SCHEMBL4864021 0.76 APP (0.73) PDE5AABCG2KMT2AMEN1MAPK1
SCHEMBL8268895 0.75 PDE5A (0.54) SIRT5PDE5AABCG2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006034512-A2 PHENYL-SUBSTITUTED QUINOLINE AND QUINAZOLINE COMPOUNDS FOR THE TREATMENT OF DIABETES BAYER PHARMACEUTICALS CORPORATION (US) 2006-03-30 WO disclosed