SCHEMBL8270102

SCHEMBL8270102

CCOC(=O)C1CCN(c2cc(-c3ccc(-c4ccccc4OCC)cc3)nc3ccccc23)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 3/20 0.54
KDM4E B2RXH2 5/20 0.53
MAPK1 P28482 3/20 0.53
SMN1; SMN2 Q16637 3/20 0.53
ALDH1A1 P00352 3/20 0.53
LMNA P02545 2/20 0.53
RAB9A P51151 2/20 0.53
NPC1 O15118 1/20 0.53
MAPT P10636 2/20 0.53
TP53 P04637 2/20 0.53
GAA P10253 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
KMT2A Q03164 3/20 0.51
MEN1 O00255 2/20 0.51
METAP1 P53582 2/20 0.47
HPGD P15428 2/20 0.47
USP2 O75604 1/20 0.47
CTNNB1 P35222 1/20 0.47
HSD17B10 Q99714 1/20 0.47
DHODH Q02127 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8268928 0.93 ALDH1A1 (0.55) KDM4EMAPK1SMN1; SMN2ALDH1A1LMNA
SCHEMBL8268926 0.91 KDM4E (0.51) PDE10AKDM4EMAPK1SMN1; SMN2ALDH1A1
SCHEMBL5794261 0.90 ALDH1A1 (0.57) PDE10AKDM4EMAPK1SMN1; SMN2ALDH1A1
SCHEMBL10992611 0.87 MAPT (0.57) KDM4EMAPK1SMN1; SMN2ALDH1A1LMNA
SCHEMBL8268364 0.83 MAPT (0.77) KDM4EMAPK1SMN1; SMN2ALDH1A1LMNA
SCHEMBL8269894 0.83 KMT2A (0.50) PDE10AKDM4ESMN1; SMN2ALDH1A1RAB9A
SCHEMBL10992499 0.81 ALDH1A1 (0.59) KDM4EMAPK1SMN1; SMN2ALDH1A1LMNA
SCHEMBL8271004 0.81 DHODH (0.61) KDM4EALDH1A1RAB9ANPC1MAPT
SCHEMBL899745 0.81 KMT2A (0.74) KDM4EALDH1A1MAPTTP53KMT2A
SCHEMBL7506358 0.80 CTSB (0.54) KDM4EMAPK1SMN1; SMN2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006034512-A2 PHENYL-SUBSTITUTED QUINOLINE AND QUINAZOLINE COMPOUNDS FOR THE TREATMENT OF DIABETES BAYER PHARMACEUTICALS CORPORATION (US) 2006-03-30 WO disclosed