SCHEMBL8274166

SCHEMBL8274166

COc1ccc(-n2nc(OCCCI)cc2C)cc1

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 19/20 0.46
LMNA P02545 1/20 0.43
HTR2B P41595 1/20 0.43
KCNH2 Q12809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL467427 0.81 SIGMAR1 (0.70) SIGMAR1HTR2BKCNH2
SCHEMBL467287 0.80 SIGMAR1 (0.71) SIGMAR1HTR2BKCNH2
SCHEMBL467139 0.79 SIGMAR1 (0.72) SIGMAR1HTR2BKCNH2
SCHEMBL467162 0.77 SIGMAR1 (0.71) SIGMAR1
SCHEMBL466999 0.77 SIGMAR1 (0.73) SIGMAR1HTR2BKCNH2
Hydrochloric Acid SCHEMBL1896508 0.76 SIGMAR1 (0.72) SIGMAR1HTR2BKCNH2
SCHEMBL1135542 0.75 SIGMAR1 (0.55) SIGMAR1HTR2BKCNH2
SCHEMBL8274194 0.75 SIGMAR1 (0.70) SIGMAR1HTR2BKCNH2
SCHEMBL23401297 0.73 LMNA (0.53) LMNA
SCHEMBL8273600 0.73 SIGMAR1 (0.70) SIGMAR1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006021462-A1 SIGMA RECEPTOR INHIBITORS LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2006-03-02 WO disclosed