SCHEMBL8280229

SCHEMBL8280229

CC1N=C(NC(=O)OC(C)(C)C)SC1c1ccnc(NCc2ccc(C(=O)O)cc2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCP P55072 1/20 0.38
NAMPT P43490 1/20 0.35
HDAC2 Q92769 3/20 0.35
HDAC1 Q13547 8/20 0.35
HDAC6 Q9UBN7 2/20 0.35
CCNE2 O96020 1/20 0.34
CCNA2 P20248 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
CCNA1 P78396 1/20 0.34
HDAC3 O15379 2/20 0.34
NCOR1 O75376 2/20 0.34
VNN1 O95497 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
PIK3CA P42336 1/20 0.34
ACACB O00763 1/20 0.33
ACACA Q13085 1/20 0.33
AURKA O14965 1/20 0.33
RPS6KB1 P23443 1/20 0.33
ACHE P22303 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8280024 0.75 VCP (0.37) VCPHDAC2HDAC1HDAC6HDAC3
SCHEMBL211981 0.74 PI4KB (0.50) VCPHDAC2HDAC1HDAC6CCNA2
SCHEMBL8279176 0.70 HDAC1 (0.61) HDAC2HDAC1HDAC6HDAC3NCOR1
SCHEMBL8280042 0.69 HDAC1 (0.62) HDAC2HDAC1HDAC6HDAC3NCOR1
SCHEMBL16408476 0.67 VCP (0.59) VCPHDAC2HDAC1HDAC6HDAC3
SCHEMBL27640625 0.65 CYP17A1 (0.46) NAMPTHDAC1HDAC6ACACBACACA
SCHEMBL133327 0.65 KMT2A (0.60) NAMPTHDAC1
SCHEMBL8280224 0.64 VCP (0.41) VCPHDAC2HDAC1HDAC6HDAC3
SCHEMBL13879810 0.64 CYP17A1 (0.55) NAMPTHDAC1HDAC6AURKARPS6KB1
SCHEMBL13879808 0.64 AURKA (0.50) NAMPTHDAC2HDAC1HDAC6HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005092899-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2005-10-06 WO disclosed