SCHEMBL8280382

SCHEMBL8280382

CN(C[C@@H](NCl)C(C)(C)C)S(C)(=O)=O

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PER2 O15055 3/20 0.33
CRY1 Q16526 3/20 0.33
CRY2 Q49AN0 3/20 0.33
MMP1 P03956 1/20 0.33
MMP2 P08253 1/20 0.33
MMP8 P22894 1/20 0.33
MMP13 P45452 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8041801 0.83 CCR6 (0.31)
SCHEMBL8281119 0.83 CCR6 (0.31)
SCHEMBL8278785 0.82 MMP1 (0.33) PER2CRY1CRY2MMP1MMP2
SCHEMBL8271464 0.81 MMP1 (0.33) PER2CRY1CRY2MMP1MMP2
SCHEMBL13251284 0.79 MMP1 (0.35) MMP1MMP2MMP8MMP13MEN1
SCHEMBL8236840 0.78 MMP1 (0.31) MMP1MMP2MMP8MMP13
SCHEMBL13272746 0.74 GAA (0.36) ALDH1A1KMT2A
SCHEMBL13686134 0.74 MMP1 (0.35) MMP1MMP2MMP8MMP13MEN1
SCHEMBL13684376 0.73 MMP1 (0.37) MMP1MMP2MMP8MMP13ALDH1A1
SCHEMBL8194462 0.72 CA1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1737821-B1 3,4-(CYCLOPENTYL)-FUSED PROLINE COMPOUNDS AS INHIBITORS OF HEPATITIS C VIRUS NS3 SERINE PROTEASE SCHERING CORP (US) 2009-08-05 EP disclosed
US-7449447-B2 Peptidomimetic NS3-serine protease inhibitors of hepatitis C virus SCHERING CORPORATION (US) 2008-11-11 US disclosed
US-7399749-B2 Substituted prolines as inhibitors of hepatitis C virus NS3 serine protease SCHERING CORPORATION (US) 2008-07-15 US disclosed
US-7342041-B2 3,4-(cyclopentyl)-fused proline compounds as inhibitors of hepatitis C virus NS3 serine protease SCHERING CORPORATION (US) 2008-03-11 US disclosed
WO-2005087730-A1 3,4-(CYCLOPENTYL)-FUSED PROLINE COMPOUNDS AS INHIBITORS OF HEPATITIS C VIRUS NS3 SERINE PROTEASE SCHERING CORPORATION (US) 2005-09-22 WO disclosed
WO-2005021584-A2 NOVEL PEPTIDOMIMETIC NS3-SERINE PROTEASE INHIBITORS OF HEPATITIS C VIRUS SCHERING CORPORATION (US) 2005-03-10 WO disclosed