SCHEMBL8280913

SCHEMBL8280913

C=C(N)Cc1ccc(C(=O)O)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
TP53 P04637 1/20 0.50
TSHR P16473 1/20 0.50
SRD5A2 P31213 4/20 0.47
F2 P00734 1/20 0.47
PLG P00747 1/20 0.47
PRSS1 P07477 1/20 0.47
PRSS2 P07478 1/20 0.47
C1S P09871 1/20 0.47
PRSS3 P35030 1/20 0.47
ANPEP P15144 1/20 0.46
ENPEP Q07075 1/20 0.46
KMT2A Q03164 2/20 0.44
CA12 O43570 4/20 0.44
CA1 P00915 4/20 0.44
CA2 P00918 4/20 0.44
CA9 Q16790 4/20 0.44
CA14 Q9ULX7 3/20 0.43
CA3 P07451 2/20 0.43
CA4 P22748 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3690716 0.83 CA2 (0.61) ALDH1A1TP53TSHRSRD5A2F2
SCHEMBL2401022 0.79 ALDH1A1 (0.57) ALDH1A1TP53TSHRSRD5A2KMT2A
SCHEMBL1063942 0.79 ALDH1A1 (0.52) ALDH1A1TP53TSHRSRD5A2F2
SCHEMBL276932 0.78 CA2 (0.62) ALDH1A1TP53TSHRSRD5A2KMT2A
Hydrochloric Acid SCHEMBL7287603 0.78 F2 (0.55) ALDH1A1TP53TSHRSRD5A2F2
SCHEMBL13037473 0.76 ALDH1A1 (0.48) ALDH1A1TP53TSHRSRD5A2F2
SCHEMBL28329860 0.76 ALDH1A1 (0.48) ALDH1A1TP53TSHRSRD5A2F2
SCHEMBL3701685 0.76 ALDH1A1 (0.48) ALDH1A1TP53TSHRSRD5A2ANPEP
SCHEMBL13381339 0.76 TSHR (0.54) ALDH1A1TP53TSHRSRD5A2POLB
SCHEMBL2733920 0.76 ALDH1A1 (0.48) ALDH1A1TP53TSHRSRD5A2F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005092899-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2005-10-06 WO disclosed
WO-2004069823-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE, INC. (CA) 2004-08-19 WO disclosed
WO-2003024448-A2 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE, INC. (CA) 2003-03-27 WO disclosed