SCHEMBL8280967

SCHEMBL8280967

CCOc1ccc(-c2nnc(C)o2)cc1Cl

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.53
MEN1 O00255 2/20 0.53
S1PR1 P21453 2/20 0.53
HPGD P15428 6/20 0.51
KDM4E B2RXH2 6/20 0.51
ALDH1A1 P00352 5/20 0.51
HSD17B10 Q99714 5/20 0.51
RAB9A P51151 5/20 0.51
NPC1 O15118 3/20 0.51
MAPK1 P28482 2/20 0.49
LMNA P02545 2/20 0.49
NPSR1 Q6W5P4 1/20 0.49
SMN1; SMN2 Q16637 3/20 0.46
LRRK2 Q5S007 1/20 0.46
TUBB4A P04350 2/20 0.44
TUBB P07437 2/20 0.44
TUBA3C P0DPH7 2/20 0.44
TUBA1B P68363 2/20 0.44
TUBA4A P68366 2/20 0.44
TUBB4B P68371 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23349276 0.82 S1PR1 (0.56) KMT2AMEN1S1PR1HPGDKDM4E
SCHEMBL19356293 0.79 S1PR1 (0.52) KMT2AMEN1S1PR1HPGDKDM4E
SCHEMBL11884342 0.78 NOTUM (0.60) HPGDKDM4EALDH1A1HSD17B10RAB9A
SCHEMBL17559462 0.77 PRMT5 (0.55) KMT2AMEN1S1PR1HPGDKDM4E
SCHEMBL12057005 0.76 S1PR1 (0.54) S1PR1HPGDKDM4EALDH1A1HSD17B10
SCHEMBL8282012 0.75 KDM4E (0.71) KMT2AMEN1HPGDKDM4EALDH1A1
SCHEMBL17559379 0.75 PRMT5 (0.53) KMT2AMEN1S1PR1HPGDKDM4E
SCHEMBL15599433 0.74 LRRK2 (0.47) HPGDKDM4EALDH1A1HSD17B10RAB9A
SCHEMBL7805208 0.74 SNCA (0.53) HPGDLMNASMN1; SMN2LRRK2NOTUM
SCHEMBL15507192 0.74 ALDH1A1 (0.50) HPGDKDM4EALDH1A1HSD17B10RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005082866-A2 SUBSTITUTED 1, 2, 4- TRIAZOLE DERIVATIVES AS OXYTOCIN ANTAGONISTS PFIZER LIMITED (GB) 2005-09-09 WO disclosed