SCHEMBL15599433

SCHEMBL15599433

Cc1nnc(-c2ccc(F)c(Cl)c2)o1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.47
MDM2 Q00987 1/20 0.47
GRIN1 Q05586 2/20 0.46
GRIN2B Q13224 2/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
TP53 P04637 2/20 0.46
TSHR P16473 1/20 0.46
HSD17B10 Q99714 1/20 0.46
NOTUM Q6P988 4/20 0.46
LMNA P02545 1/20 0.45
HPGD P15428 1/20 0.45
KDM4E B2RXH2 1/20 0.44
GSK3B P49841 2/20 0.41
MAPK14 Q16539 1/20 0.41
RPA1 P27694 1/20 0.41
GPR84 Q9NQS5 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11884342 0.84 NOTUM (0.60) LRRK2SMN1; SMN2NPC1RAB9AHSD17B10
SCHEMBL26766195 0.84 NOTUM (0.49) GRIN1GRIN2BSMN1; SMN2NPC1RAB9A
SCHEMBL8415605 0.83 NOTUM (0.48) GRIN1GRIN2BSMN1; SMN2NPC1RAB9A
SCHEMBL8229635 0.80 NOTUM (0.46) SMN1; SMN2NPC1RAB9ATP53TSHR
SCHEMBL7805208 0.80 SNCA (0.53) LRRK2SMN1; SMN2NOTUMLMNAHPGD
SCHEMBL18567895 0.80 NOTUM (0.46) SMN1; SMN2NPC1RAB9ATP53TSHR
SCHEMBL15507192 0.80 ALDH1A1 (0.50) LRRK2SMN1; SMN2NPC1RAB9ATP53
SCHEMBL13451187 0.80 NOTUM (0.46) SMN1; SMN2NPC1RAB9ATP53HSD17B10
SCHEMBL14932735 0.79 NOTUM (0.48) SMN1; SMN2NPC1RAB9ANOTUMLMNA
SCHEMBL2310162 0.78 NPC1 (0.60) SMN1; SMN2NPC1RAB9ATP53TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9505749-B2 Quinazolinone compounds and derivatives thereof AMGEN INC. (US) 2016-11-29 US disclosed
US-20150225396-A1 Quinazolinone Compounds and Derivatives Thereof AMGEN INC. 2015-08-13 US disclosed
WO-2014036022-A1 QUINAZOLINONE COMPOUNDS AND DERIVATIVES THEREOF AMGEN INC. (US) 2014-03-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150225396-A1 Quinazolinone Compounds and Derivatives Thereof TNKS, TPI1, TNKS1BP1 LRRK2 1351/4885MDM2 717/4885GRIN1 3245/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.