SCHEMBL8281024

SCHEMBL8281024

CCOCc1nnc(-c2ccc(O[C@@H](C)COC)cc2)n1-c1ccc(OC)nc1

nearest known ligand 0.62

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
OXTR P30559 18/20 0.62
AVPR1A P37288 16/20 0.62
AVPR2 P30518 8/20 0.58
AVPR1B P47901 3/20 0.39
KCNH2 Q12809 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8281748 1.00 OXTR (0.62) OXTRAVPR1AAVPR2AVPR1BKCNH2
SCHEMBL8279852 0.93 OXTR (0.63) OXTRAVPR1AAVPR2
SCHEMBL8281026 0.93 OXTR (0.63) OXTRAVPR1AAVPR2
SCHEMBL8279850 0.90 OXTR (0.55) OXTRAVPR1AAVPR2
SCHEMBL8282612 0.90 OXTR (0.55) OXTRAVPR1AAVPR2
SCHEMBL8281643 0.87 OXTR (0.52) OXTRAVPR1AAVPR2
SCHEMBL8282002 0.87 OXTR (0.52) OXTRAVPR1AAVPR2
SCHEMBL8282551 0.87 OXTR (0.54) OXTRAVPR1AAVPR2
SCHEMBL8279860 0.86 OXTR (0.50) OXTRAVPR1AAVPR2
SCHEMBL8281687 0.83 OXTR (0.48) OXTRAVPR1AAVPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005082866-A2 SUBSTITUTED 1, 2, 4- TRIAZOLE DERIVATIVES AS OXYTOCIN ANTAGONISTS PFIZER LIMITED (GB) 2005-09-09 WO disclosed