SCHEMBL8281137

SCHEMBL8281137

Cc1cc(C(O)CF)ccc1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 4/20 0.45
ADRA2B P18089 4/20 0.45
ADRA2C P18825 4/20 0.45
ADRB1 P08588 3/20 0.45
ADRB3 P13945 3/20 0.45
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
MEN1 O00255 3/20 0.33
MAPT P10636 3/20 0.33
KMT2A Q03164 3/20 0.33
TDP1 Q9NUW8 3/20 0.33
ADRB2 P07550 3/20 0.33
KDM4E B2RXH2 2/20 0.33
ADORA3 P0DMS8 2/20 0.33
DRD2 P14416 2/20 0.33
DRD1 P21728 2/20 0.33
ADRA1D P25100 2/20 0.33
ADRA1A P35348 2/20 0.33
PTGS2 P35354 2/20 0.33
ADRA1B P35368 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17947385 0.85 LMNA (0.45) ADRA2AADRA2BADRA2CADRB1ADRB3
SCHEMBL8257922 0.85 LMNA (0.45) ADRA2AADRA2BADRA2CADRB1ADRB3
SCHEMBL13862134 0.85 CYP3A4 (0.46) ADRA2AADRA2BADRA2CADRB1ADRB3
SCHEMBL15787308 0.81 ADRB1 (0.42) ADRA2AADRA2BADRA2CADRB1ADRB3
SCHEMBL15787309 0.81 ADRB1 (0.42) ADRA2AADRA2BADRA2CADRB1ADRB3
SCHEMBL8251464 0.78 UGT2B7 (0.45) ADRA2AADRA2BADRA2CADRB1ADRB3
SCHEMBL16956357 0.77 DAO (0.33) ADRA2AADRA2BADRA2CADRB1ADRB3
SCHEMBL639301 0.76 AKR1C3 (0.40) ADRA2AADRA2BADRA2CADRB1ADRB3
SCHEMBL639829 0.76 AKR1C3 (0.40) ADRA2AADRA2BADRA2CADRB1ADRB3
SCHEMBL10178370 0.76 ADRB1 (0.39) ADRA2AADRA2BADRA2CADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005103055-A1 PYRAZOLO-[4,3-e]-1,2,4-TRIAZOLO-[1,5-c]-PYRIMIDINE ADENOSINE A2A RECEPTOR ANTAGONISTS SCHERING CORPORATION (US) 2005-11-03 WO disclosed