SCHEMBL8282942

SCHEMBL8282942

CO[n+]1ccc2c(c1)C(=O)N(C[C@@H](NC(=O)OC(C)(C)C)C(C)(C)C)C2=O

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.33
GLA P06280 2/20 0.33
GAA P10253 2/20 0.33
MAPT P10636 2/20 0.33
PPARG P37231 2/20 0.33
PPARA Q07869 2/20 0.33
BRD4 O60885 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA7 P43166 2/20 0.33
CA4 P22748 1/20 0.33
CA9 Q16790 1/20 0.33
ATM Q13315 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
RORC P51449 1/20 0.33
AKT1 P31749 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8282957 0.83 ALDH1A1 (0.43) MAPTPPARGPPARAALDH1A1CA9
SCHEMBL8178666 0.83 ALDH1A1 (0.43) MAPTPPARGPPARAALDH1A1CA9
SCHEMBL13622642 0.83 ALDH1A1 (0.43) MAPTPPARGPPARAALDH1A1CA9
SCHEMBL8282944 0.77 NPSR1 (0.44) KDM4EGAAMAPTALDH1A1TSHR
SCHEMBL13622658 0.77 NPSR1 (0.44) KDM4EGAAMAPTALDH1A1TSHR
SCHEMBL12679223 0.72 CTSS (0.43) PPARGPPARAALDH1A1CA9ATM
SCHEMBL3387424 0.71 ALDH1A1 (0.43) MAPTALDH1A1ATMCTSSCTSK
SCHEMBL13622704 0.71 KMT2A (0.43) GAAMAPTALDH1A1HSD17B10ATM
SCHEMBL13632866 0.71 KMT2A (0.43) GAAMAPTALDH1A1HSD17B10ATM
SCHEMBL5551909 0.70 CA1 (0.50) ALDH1A1CA1CA2CA7CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730142-B1 NOVEL KETOAMIDES WITH CYCLIC P4'S AS INHIBITORS OF NS3 SERINE PROTEASE OF HEPATITIS C VIRUS SCHERING CORP (US) 2011-06-29 EP disclosed
WO-2005085242-A1 NOVEL KETOAMIDES WITH CYCLIC P4'S AS INHIBITORS OF NS3 SERINE PROTEASE OF HEPATITIS C VIRUS SCHERING CORPORATION (US) 2005-09-15 WO disclosed