SCHEMBL8283586

SCHEMBL8283586

C=C(C)C[C@H]1OCCN(C(=O)OCc2ccccc2)[C@@H]1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
PREP P48147 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
SIGMAR1 Q99720 1/20 0.43
AGTR2 P50052 2/20 0.42
FKBP1A P62942 1/20 0.41
ELANE P08246 1/20 0.41
HTR2C P28335 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8355480 0.81 ELANE (0.49) NPC1RAB9ASMN1; SMN2SIGMAR1AGTR2
SCHEMBL8281753 0.81 ELANE (0.49) NPC1RAB9ASMN1; SMN2SIGMAR1AGTR2
SCHEMBL6358373 0.77 PREP (0.57) MEN1KMT2ANPSR1PREPNPC1
SCHEMBL6105877 0.77 PREP (0.57) MEN1KMT2ANPSR1PREPNPC1
SCHEMBL16256991 0.76 MEN1 (0.49) MEN1KMT2ANPSR1PREPNPC1
SCHEMBL14546519 0.76 AGTR2 (0.46) NPC1RAB9ASMN1; SMN2SIGMAR1AGTR2
SCHEMBL8279476 0.76 ELANE (0.44) NPC1RAB9ASMN1; SMN2AGTR2FKBP1A
SCHEMBL10137614 0.76 ELANE (0.44) NPC1RAB9ASMN1; SMN2AGTR2FKBP1A
SCHEMBL8280446 0.76 AGTR2 (0.46) NPC1RAB9ASMN1; SMN2SIGMAR1AGTR2
SCHEMBL14569818 0.76 AGTR2 (0.46) NPC1RAB9ASMN1; SMN2SIGMAR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730142-B1 NOVEL KETOAMIDES WITH CYCLIC P4'S AS INHIBITORS OF NS3 SERINE PROTEASE OF HEPATITIS C VIRUS SCHERING CORP (US) 2011-06-29 EP disclosed
WO-2005085197-A1 CYCLOBUTENEDIONE GROUPS-CONTAINING COMPOUNDS AS INHIBITORS OF HEPATITIS C VIRUS NS3 SERINE PROTEASE SCHERING CORPORATION (US) 2005-09-15 WO disclosed