SCHEMBL8285169

SCHEMBL8285169

Cc1cc(C(=O)c2ccccc2)nc2c1c(=O)cc(Nc1ccccc1)n2-c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE11A Q9HCR9 1/20 0.45
ALDH1A1 P00352 3/20 0.43
MAPT P10636 5/20 0.40
GAA P10253 3/20 0.38
GFER P55789 1/20 0.38
POLB P06746 3/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
HTT P42858 2/20 0.37
HPGD P15428 2/20 0.36
MAPK1 P28482 1/20 0.36
MAPK13 O15264 1/20 0.35
MAPK12 P53778 1/20 0.35
MAPK11 Q15759 1/20 0.35
MAPK14 Q16539 1/20 0.35
KDM4E B2RXH2 2/20 0.35
MEN1 O00255 1/20 0.35
TP53 P04637 1/20 0.35
ALOX15 P16050 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8285193 0.93 PDE11A (0.44) PDE11AALDH1A1MAPTGAAGFER
SCHEMBL8285205 0.93 MAPT (0.44) PDE11AALDH1A1MAPTGAAGFER
SCHEMBL8285220 0.91 PDE11A (0.43) PDE11AALDH1A1MAPTPOLBNPC1
SCHEMBL5872175 0.90 PDE11A (0.47) PDE11AALDH1A1MAPTGAAGFER
SCHEMBL5871541 0.89 PDE11A (0.46) PDE11AALDH1A1MAPTGAAGFER
SCHEMBL8287397 0.88 PDE11A (0.46) PDE11AALDH1A1MAPTGAAGFER
SCHEMBL8287393 0.88 PDE11A (0.46) PDE11AALDH1A1MAPTPOLBNPC1
SCHEMBL8287518 0.86 PDE11A (0.44) PDE11AALDH1A1MAPTGAAGFER
SCHEMBL8285223 0.86 PDE11A (0.44) PDE11AALDH1A1MAPTGAAGFER
SCHEMBL8285216 0.86 PDE11A (0.43) PDE11AALDH1A1MAPTGAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005091857-A2 1,6-NAPHTHYRIDINE AND 1,8-NAPHTHYRIDINE DERIVATIVES AND THEIR USE TO TREAT DIABETES AND RELATED DISORDERS BAYER PHARMACEUTICALS CORPORATION (US) 2005-10-06 WO disclosed
WO-2003027112-A1 1, 8-NAPHTHYRIDINE DERIVATIVES AS ANTIDIABETICS BAYER PHARMACEUTICALS CORPORATION (US) 2003-04-03 WO disclosed