SCHEMBL8285208

SCHEMBL8285208

Cc1nc2c(cc1CCC(=O)N(C)C)c(=O)cc(Nc1ccccc1)n2-c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAT2A P31153 2/20 0.38
PDE11A Q9HCR9 1/20 0.38
CSF1R P07333 1/20 0.35
NR4A1 P22736 1/20 0.34
NR4A2 P43354 1/20 0.34
NR4A3 Q92570 1/20 0.34
KDM4E B2RXH2 1/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MAPT P10636 1/20 0.34
FFAR1 O14842 1/20 0.33
P2RX7 Q99572 1/20 0.33
RXRA P19793 1/20 0.33
GAA P10253 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
GFER P55789 1/20 0.32
HPGD P15428 1/20 0.32
MAPK1 P28482 1/20 0.32
TP53 P04637 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5911507 0.90 PLA2G4A (0.40) PDE11ACSF1RKDM4EHTTMAPT
SCHEMBL8285190 0.89 PDE11A (0.39) PDE11ACSF1RKDM4EHTTMAPT
SCHEMBL8287111 0.89 PDE11A (0.39) PDE11ACSF1RMAPTGAAMEN1
SCHEMBL8287185 0.88 PDE11A (0.38) PDE11ACSF1RMAPTRXRAGAA
SCHEMBL8287884 0.88 TP53 (0.44) KDM4EHTTMAPTGAAKMT2A
SCHEMBL8285207 0.88 PDE11A (0.38) MAT2APDE11ANR4A2MAPTGAA
SCHEMBL8285219 0.85 PDE11A (0.39) PDE11AKDM4EHTTNPSR1GAA
SCHEMBL8287927 0.84 NPC1 (0.41) PDE11AKDM4EMAPTGAAKMT2A
SCHEMBL8287150 0.84 PDE11A (0.40) PDE11ACSF1RKDM4EHTTNPSR1
SCHEMBL8285235 0.84 PDE11A (0.41) MAT2APDE11ACSF1RKDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005091857-A2 1,6-NAPHTHYRIDINE AND 1,8-NAPHTHYRIDINE DERIVATIVES AND THEIR USE TO TREAT DIABETES AND RELATED DISORDERS BAYER PHARMACEUTICALS CORPORATION (US) 2005-10-06 WO disclosed
WO-2003027112-A1 1, 8-NAPHTHYRIDINE DERIVATIVES AS ANTIDIABETICS BAYER PHARMACEUTICALS CORPORATION (US) 2003-04-03 WO disclosed