SCHEMBL8288013

SCHEMBL8288013

CC(C)(C)OC(=O)NC1CCN(C(=O)c2ccc(Cl)s2)C1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.48
HSD11B1 P28845 3/20 0.47
CYP2C9 P11712 1/20 0.47
ALDH1A1 P00352 1/20 0.47
HPGD P15428 1/20 0.47
ADORA2A P29274 7/20 0.47
ADORA2B P29275 5/20 0.47
ADORA3 P0DMS8 2/20 0.47
CTSK P43235 2/20 0.46
HDAC3 O15379 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC2 Q92769 1/20 0.46
F10 P00742 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CFTR P13569 1/20 0.45
NAMPT P43490 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3449128 0.82 USP30 (0.55) PARP1ALDH1A1ADORA2AADORA2BADORA3
SCHEMBL3449130 0.82 USP30 (0.55) PARP1ALDH1A1ADORA2AADORA2BADORA3
SCHEMBL6371116 0.82 ALDH1A1 (0.55) ALDH1A1HPGDF10CA1CA2
SCHEMBL6310345 0.78 CFTR (0.48) PARP1HSD11B1CYP2C9ADORA2AADORA2B
SCHEMBL2610266 0.78 NAMPT (0.61) PARP1HSD11B1CYP2C9CTSKHDAC3
SCHEMBL7939466 0.78 NAMPT (0.61) PARP1HSD11B1CYP2C9CTSKHDAC3
SCHEMBL31222941 0.78 HSD11B1 (0.45) PARP1HSD11B1CYP2C9ADORA2AADORA2B
SCHEMBL24185654 0.77 EPHX2 (0.52) PARP1HSD11B1CYP2C9ADORA2AADORA2B
SCHEMBL31267054 0.77 NAMPT (0.57) PARP1HSD11B1CYP2C9ADORA2AADORA2B
SCHEMBL31267093 0.77 NAMPT (0.57) PARP1HSD11B1CYP2C9ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005032472-A2 PYRROLIDINE AND PIPERIDINE DERIVATIVES AS FACTOR XA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-04-14 WO disclosed