SCHEMBL8288556

SCHEMBL8288556

CCC(C)(C)C1CCc2c(sc(NC(=O)c3cccnc3)c2C#N)C1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 9/20 0.69
NPSR1 Q6W5P4 1/20 0.69
SAE1 Q9UBE0 1/20 0.69
UBA2 Q9UBT2 1/20 0.69
GCGR P47871 1/20 0.65
LMNA P02545 5/20 0.64
GAA P10253 2/20 0.64
ALDH1A1 P00352 7/20 0.54
KDM4E B2RXH2 5/20 0.54
RAB9A P51151 2/20 0.54
HPGD P15428 5/20 0.52
SMN1; SMN2 Q16637 4/20 0.52
HSD17B10 Q99714 2/20 0.51
THRB P10828 1/20 0.49
HTT P42858 1/20 0.49
POLB P06746 5/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
ALOX15 P16050 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8289724 0.87 ALDH1A1 (0.59) MAPTNPSR1SAE1UBA2GCGR
SCHEMBL16689136 0.85 GCGR (0.66) MAPTNPSR1SAE1UBA2GCGR
SCHEMBL2649274 0.79 GCGR (0.76) MAPTNPSR1SAE1UBA2GCGR
SCHEMBL2647850 0.79 GCGR (1.00) MAPTNPSR1SAE1UBA2GCGR
SCHEMBL31075000 0.78 MAPT (0.96) MAPTLMNAGAAALDH1A1KDM4E
SCHEMBL2648864 0.78 GCGR (0.74) MAPTNPSR1SAE1UBA2GCGR
SCHEMBL2647883 0.78 GCGR (0.73) MAPTNPSR1SAE1UBA2GCGR
SCHEMBL3282241 0.78 MAPT (0.71) MAPTNPSR1SAE1UBA2GCGR
SCHEMBL13210588 0.78 HPGD (0.68) MAPTNPSR1SAE1UBA2GCGR
SCHEMBL2648446 0.77 MAPT (0.71) MAPTNPSR1SAE1UBA2GCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed