SCHEMBL8288674

SCHEMBL8288674

CC(C)(C)CC(=O)Nc1sc2c(c1C(N)=O)CCCC2

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 4/20 0.74
KDM4E B2RXH2 2/20 0.70
MAPK1 P28482 1/20 0.70
ANO1 Q5XXA6 1/20 0.68
ALDH1A1 P00352 5/20 0.67
TSHR P16473 4/20 0.67
LMNA P02545 3/20 0.67
MEN1 O00255 2/20 0.67
KMT2A Q03164 2/20 0.67
MAPT P10636 2/20 0.67
CYP1A2 P05177 1/20 0.67
CYP2C19 P33261 1/20 0.67
GFER P55789 1/20 0.67
L3MBTL1 Q9Y468 1/20 0.67
CNR1 P21554 4/20 0.66
CNR2 P34972 4/20 0.66
HPGD P15428 4/20 0.64
GAA P10253 1/20 0.64
RAB9A P51151 1/20 0.64
MAPK10 P53779 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8288772 0.97 KDM4E (0.74) FLT3KDM4EMAPK1ANO1ALDH1A1
SCHEMBL5453467 0.85 FLT3 (1.00) FLT3KDM4EMAPK1ANO1ALDH1A1
SCHEMBL14513178 0.83 ALDH1A1 (0.69) KDM4EMAPK1ALDH1A1TSHRLMNA
SCHEMBL5465217 0.83 ALDH1A1 (0.81) FLT3KDM4EMAPK1ANO1ALDH1A1
SCHEMBL5455157 0.83 CNR2 (0.69) FLT3KDM4EMAPK1ANO1ALDH1A1
SCHEMBL8289709 0.83 MAPT (0.69) KDM4EMAPK1ANO1ALDH1A1MEN1
SCHEMBL8289412 0.82 KDM4E (1.00) FLT3KDM4EMAPK1ALDH1A1TSHR
SCHEMBL3924390 0.82 ANO1 (0.97) FLT3KDM4EMAPK1ANO1ALDH1A1
SCHEMBL3453042 0.82 FLT3 (0.75) FLT3KDM4EMAPK1ANO1ALDH1A1
SCHEMBL4135422 0.82 HPGD (0.83) FLT3KDM4EMAPK1ANO1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed