SCHEMBL8289727

SCHEMBL8289727

COC(=O)c1c(NC(=O)CCCC(=O)O)sc2c1CCC(c1ccccc1)C2

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.63
KDM4E B2RXH2 5/20 0.63
MAPT P10636 7/20 0.62
POLB P06746 3/20 0.53
KMT2A Q03164 1/20 0.52
HSD17B10 Q99714 3/20 0.52
ALOX15 P16050 2/20 0.52
HPGD P15428 2/20 0.52
RAB9A P51151 2/20 0.52
ALOX12 P18054 1/20 0.52
MAPK1 P28482 1/20 0.52
TP53 P04637 2/20 0.49
NPC1 O15118 1/20 0.49
AIP O00170 1/20 0.48
SGTA O43765 1/20 0.48
TOMM70 O94826 1/20 0.48
STIP1 P31948 1/20 0.48
PPP5C P53041 1/20 0.48
DNAJC7 Q99615 1/20 0.48
STUB1 Q9UNE7 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5371517 0.85 ALDH1A1 (0.56) ALDH1A1KDM4EMAPTPOLBHSD17B10
SCHEMBL918839 0.81 ALDH1A1 (0.67) ALDH1A1KDM4EMAPTPOLBKMT2A
SCHEMBL21247397 0.80 TP53 (0.60) ALDH1A1KDM4EMAPTPOLBKMT2A
SCHEMBL21250170 0.77 TP53 (0.54) ALDH1A1KDM4EMAPTPOLBHSD17B10
SCHEMBL4227925 0.77 MAPT (0.48) ALDH1A1KDM4EMAPTPOLBKMT2A
SCHEMBL7929684 0.75 PDE4B (0.55) ALDH1A1MAPTPOLBKMT2AHPGD
SCHEMBL918266 0.75 POLB (0.64) ALDH1A1KDM4EMAPTPOLBHSD17B10
SCHEMBL6204554 0.75 ALDH1A1 (0.61) ALDH1A1KDM4EMAPTKMT2AHSD17B10
SCHEMBL21260713 0.72 PDE4B (0.52) ALDH1A1MAPTPOLBKMT2AHSD17B10
SCHEMBL21260738 0.72 MAPT (0.54) ALDH1A1KDM4EMAPTPOLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed