SCHEMBL8289768

SCHEMBL8289768

COC(=O)c1c(NC(=O)CSc2nnc(-c3ccc(O)cc3)o2)sc(C(C)=O)c1C

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.78
HPGD P15428 4/20 0.75
ALDH1A1 P00352 4/20 0.75
TSHR P16473 6/20 0.67
KMT2A Q03164 3/20 0.67
MAPK1 P28482 2/20 0.67
USP2 O75604 4/20 0.64
MEN1 O00255 2/20 0.64
FKBP4 Q02790 1/20 0.58
FKBP5 Q13451 1/20 0.58
MAPT P10636 3/20 0.57
PKM P14618 3/20 0.55
HSD17B10 Q99714 2/20 0.55
POLB P06746 1/20 0.55
PPARG P37231 1/20 0.55
NCOA2 Q15596 1/20 0.55
NCOA1 Q15788 1/20 0.55
NPC1 O15118 4/20 0.55
RAB9A P51151 3/20 0.55
SMN1; SMN2 Q16637 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19635942 0.73 ALDH1A1 (0.68) NPSR1HPGDALDH1A1TSHRKMT2A
SCHEMBL16208829 0.71 TSHR (0.67) NPSR1HPGDALDH1A1TSHRKMT2A
SCHEMBL10016415 0.68 NPC1 (1.00) NPSR1ALDH1A1TSHRKMT2AMAPT
SCHEMBL21104909 0.68 ALDH1A1 (1.00) NPSR1HPGDALDH1A1TSHRKMT2A
SCHEMBL17068788 0.67 HSP90AA1 (0.74) NPSR1HPGDALDH1A1TSHRMAPK1
SCHEMBL8289563 0.67 ALDH1A1 (0.84) NPSR1HPGDALDH1A1TSHRKMT2A
SCHEMBL13167282 0.66 TP53 (1.00) NPSR1ALDH1A1TSHRMAPK1MAPT
SCHEMBL243554 0.66 CA12 (0.74) KMT2AUSP2MEN1MAPTPKM
SCHEMBL10016428 0.64 TP53 (0.80) NPSR1HPGDALDH1A1TSHRKMT2A
SCHEMBL21447020 0.63 RAB9A (0.64) ALDH1A1TSHRMAPTPKMHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed