SCHEMBL8289840

SCHEMBL8289840

NC(=O)c1c(NC(=O)c2ccc(Cl)cc2Cl)sc2c1CCCCC2

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.77
RAB9A P51151 7/20 0.77
CFTR P13569 1/20 0.76
FLT3 P36888 9/20 0.69
HPGD P15428 2/20 0.64
ALDH1A1 P00352 3/20 0.62
SMN1; SMN2 Q16637 3/20 0.62
KDM4E B2RXH2 2/20 0.62
LMNA P02545 2/20 0.62
ALOX15 P16050 2/20 0.62
TSHR P16473 2/20 0.62
HSD17B10 Q99714 2/20 0.62
MAPT P10636 2/20 0.62
KMT2A Q03164 3/20 0.60
MEN1 O00255 2/20 0.60
POLB P06746 1/20 0.60
TNF P01375 1/20 0.60
NOD1 Q9Y239 1/20 0.60
ESR1 P03372 1/20 0.59
TP53 P04637 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8290644 0.89 NPC1 (0.96) NPC1RAB9ACFTRFLT3HPGD
SCHEMBL8290776 0.87 NPC1 (1.00) NPC1RAB9ACFTRFLT3HPGD
SCHEMBL3110880 0.86 CFTR (1.00) NPC1RAB9ACFTRFLT3HPGD
SCHEMBL4138685 0.84 MAPT (0.75) NPC1RAB9ACFTRFLT3ALDH1A1
SCHEMBL8290832 0.84 NPC1 (1.00) NPC1RAB9ACFTRFLT3HPGD
SCHEMBL8289853 0.83 FLT3 (0.97) NPC1RAB9ACFTRFLT3ALDH1A1
SCHEMBL8290663 0.82 FLT3 (1.00) NPC1RAB9ACFTRFLT3ALDH1A1
SCHEMBL8289839 0.82 FLT3 (0.98) NPC1RAB9ACFTRFLT3ALDH1A1
SCHEMBL3282296 0.81 TP53 (0.71) NPC1RAB9AHPGDALDH1A1SMN1; SMN2
SCHEMBL8288686 0.81 FLT3 (1.00) NPC1RAB9ACFTRFLT3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed