SCHEMBL8290776

SCHEMBL8290776

NC(=O)c1c(NC(=O)c2ccc(F)cc2Cl)sc2c1CCC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 1.00
RAB9A P51151 6/20 1.00
CFTR P13569 1/20 0.69
FLT3 P36888 4/20 0.60
MAPT P10636 4/20 0.60
ANO1 Q5XXA6 1/20 0.59
HPGD P15428 3/20 0.59
KMT2A Q03164 5/20 0.58
MEN1 O00255 4/20 0.58
CASP3 P42574 1/20 0.58
SENP7 Q9BQF6 1/20 0.58
L3MBTL1 Q9Y468 3/20 0.58
ALDH1A1 P00352 2/20 0.56
GAA P10253 2/20 0.56
KDM4E B2RXH2 2/20 0.56
LMNA P02545 1/20 0.56
TNF P01375 1/20 0.55
NOD1 Q9Y239 1/20 0.55
HTT P42858 1/20 0.55
NPSR1 Q6W5P4 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8290644 0.98 NPC1 (0.96) NPC1RAB9ACFTRFLT3MAPT
SCHEMBL8289840 0.87 NPC1 (0.77) NPC1RAB9ACFTRFLT3MAPT
SCHEMBL8290832 0.84 NPC1 (1.00) NPC1RAB9ACFTRFLT3ANO1
SCHEMBL3110880 0.82 CFTR (1.00) NPC1RAB9ACFTRFLT3ANO1
SCHEMBL8289526 0.79 RAB9A (0.95) NPC1RAB9AFLT3MAPTKMT2A
SCHEMBL8288827 0.79 HPGD (0.71) NPC1RAB9ACFTRFLT3MAPT
SCHEMBL8288680 0.79 NPC1 (0.67) NPC1RAB9ACFTRFLT3MAPT
SCHEMBL8289720 0.78 NPC1 (0.73) NPC1RAB9ACFTRFLT3MAPT
SCHEMBL8289437 0.78 FLT3 (0.95) NPC1RAB9ACFTRFLT3MAPT
SCHEMBL8288830 0.77 NPC1 (0.64) NPC1RAB9ACFTRFLT3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed