SCHEMBL8289934

SCHEMBL8289934

Cc1ccc2c(c1C)C(N)=NC2

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.38
HTR5A P47898 5/20 0.36
NOS3 P29474 2/20 0.33
NOS2 P35228 2/20 0.33
TDP2 O95551 1/20 0.33
NSD2 O96028 1/20 0.33
HSP90AA1 P07900 1/20 0.33
PAX8 Q06710 1/20 0.33
AKT1 P31749 1/20 0.32
AKT2 P31751 1/20 0.32
AKT3 Q9Y243 1/20 0.32
POLB P06746 1/20 0.31
NOS1 P29475 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10198725 0.78 HTR5A (0.53) TSHRHTR5ANOS3NOS2PAX8
SCHEMBL15313038 0.67 TDP2 (0.52) TSHRNOS3NOS2TDP2NSD2
SCHEMBL8267504 0.64 TSHR (0.52) TSHRHTR5A
SCHEMBL9949264 0.64 HTR5A (0.51) TSHRHTR5ANOS3NOS2NOS1
SCHEMBL30238157 0.63 TDP2 (0.44) TSHRNOS3NOS2TDP2NSD2
SCHEMBL3215787 0.63 TDP2 (0.44) TSHRNOS3NOS2TDP2NSD2
SCHEMBL10158893 0.61
SCHEMBL8269241 0.60 TSHR (0.52) TSHRHTR5ANOS3NOS2POLB
SCHEMBL4014088 0.58 TDP2 (0.45) TDP2NSD2HSP90AA1PAX8AKT1
SCHEMBL9854240 0.58 TDP2 (0.44) TSHRNOS3NOS2TDP2NSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005032490-A2 CYCLIC DIAMINES AND DERIVATIVES AS FACTOR XA INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-04-14 WO disclosed