SCHEMBL8290122

SCHEMBL8290122

Cn1c(-c2ccccc2)nc(N2CCCCC2)c(Oc2ccccc2C#N)c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.43
ALDH1A1 P00352 7/20 0.43
HPGD P15428 5/20 0.43
L3MBTL1 Q9Y468 3/20 0.43
LMNA P02545 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
DCK P27707 3/20 0.40
ADORA2A P29274 2/20 0.39
TSHR P16473 3/20 0.38
HSD17B10 Q99714 2/20 0.38
MAPT P10636 2/20 0.38
NPY5R Q15761 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
KDM5A P29375 1/20 0.37
USP2 O75604 1/20 0.37
TP53 P04637 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13139852 0.88 DPP4 (0.50) DPP4
SCHEMBL3064302 0.88 DPP4 (0.50) DPP4
SCHEMBL8290105 0.84 KDM4E (0.44) KDM4EALDH1A1HPGDL3MBTL1LMNA
SCHEMBL14238617 0.82 POLB (0.43) KDM4EALDH1A1HPGDLMNAADORA2A
SCHEMBL5583740 0.81 PIN1 (0.40) KDM4EALDH1A1HPGDL3MBTL1LMNA
SCHEMBL8290094 0.78 DPP4 (0.44) KDM4EALDH1A1HPGDL3MBTL1LMNA
SCHEMBL8291764 0.75 ALDH1A1 (0.42) KDM4EALDH1A1HPGDL3MBTL1LMNA
SCHEMBL13139855 0.73 DPP4 (0.57) DPP4
SCHEMBL3075383 0.73 DPP4 (0.57) DPP4
SCHEMBL5369275 0.67 NPY5R (0.50) KDM4EALDH1A1HPGDADORA2ANPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1699777-B1 DIPEPTIDYL PEPTIDASE INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2012-12-12 EP disclosed
WO-2005026148-A1 DIPEPTIDYL PEPTIDASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2005-03-24 WO disclosed