SCHEMBL8290900

SCHEMBL8290900

Clc1ccc(C2(CCCOC3CCCCO3)CCCNC2)cc1Cl

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 19/20 0.55
SLC6A3 Q01959 18/20 0.55
SLC6A2 P23975 16/20 0.55
CYP2D6 P10635 2/20 0.52
CYP1A1 P04798 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7751548 0.97 SLC6A4 (0.56) SLC6A4SLC6A3SLC6A2CYP2D6CYP1A1
SCHEMBL7947168 0.95 SLC6A2 (0.48) SLC6A4SLC6A3SLC6A2CYP2D6CYP1A1
SCHEMBL7077339 0.94 SLC6A4 (0.57) SLC6A4SLC6A3SLC6A2CYP2D6CYP1A1
SCHEMBL8452305 0.91 SLC6A4 (0.58) SLC6A4SLC6A3SLC6A2CYP2D6CYP1A1
SCHEMBL6957304 0.89 SLC6A2 (0.50) SLC6A4SLC6A3SLC6A2CYP2D6CYP1A1
SCHEMBL6544366 0.85 SLC6A3 (0.38) SLC6A4SLC6A3SLC6A2CYP2D6
SCHEMBL8291781 0.84 SLC6A3 (0.46) SLC6A4SLC6A3SLC6A2CYP2D6CYP1A1
SCHEMBL7091052 0.84 SLC6A4 (0.57) SLC6A4SLC6A3SLC6A2CYP2D6CYP3A4
SCHEMBL7764201 0.84 TACR1 (0.40) SLC6A4SLC6A3SLC6A2CYP2D6
SCHEMBL7956526 0.82 MEN1 (0.38) SLC6A4SLC6A3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0512901-B1 Aminated polycyclic compounds and their enantiomers, process for their preparation and pharmaceutical compositions containing them SANOFI SA (FR) 1999-06-23 EP claimed
US-5770735-A Polycyclic amine compounds and their enantiomers, their method of preparation and pharmaceutical compositions in which they are present ELF SANOFI (FR) 1998-06-23 US claimed
EP-0512901-B1 Aminated polycyclic compounds and their enantiomers, process for their preparation and pharmaceutical compositions containing them SANOFI SA (FR) 1999-06-23 EP disclosed
US-5770735-A Polycyclic amine compounds and their enantiomers, their method of preparation and pharmaceutical compositions in which they are present ELF SANOFI (FR) 1998-06-23 US disclosed
US-5625060-A Polycyclic amine compounds and their enantiomers, their method of preparation and pharmaceutical compositions on which they are present Sanofi, Elf (FR) 1997-04-29 US disclosed
US-5340822-A Substance P, neurokinin antagonists ELF SANOFI (FR) 1994-08-23 US disclosed
EP-0512901-A1 Aminated polycyclic compounds and their enantiomers, process for their preparation and pharmaceutical compositions containing them SANOFI (FR) 1992-11-11 EP disclosed