SCHEMBL8292256

SCHEMBL8292256

O=c1[nH]c(=O)n([C@@H]2CO[C@H](CO)[C@@H](O)C2)cc1/C=C/Br

nearest known ligand 0.70

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TK1 P04183 5/20 0.70
CYP1A2 P05177 1/20 0.70
CYP3A4 P08684 1/20 0.70
TSHR P16473 1/20 0.70
BLM P54132 1/20 0.70
PMP22 Q01453 1/20 0.70
NPSR1 Q6W5P4 1/20 0.70
TK2 O00142 8/20 0.60
LMNA P02545 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1469836 0.83 TK1 (0.67) TK1CYP1A2CYP3A4TSHRBLM
SCHEMBL1469838 0.83 TK1 (0.67) TK1CYP1A2CYP3A4TSHRBLM
SCHEMBL4977332 0.83 TK1 (0.67) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL5983819 0.82 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL1172398 0.82 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL4283382 0.82 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL141407 0.82 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL21316784 0.82 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL4283383 0.82 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL13674189 0.82 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0608809-B1 Antiviral tetrahydropyrans BRISTOL MYERS SQUIBB CO (US) 1999-07-07 EP claimed
EP-0608809-A1 Antiviral tetrahydropyrans BRISTOL-MYERS SQUIBB COMPANY (US) 1994-08-03 EP claimed
EP-0608809-B1 Antiviral tetrahydropyrans BRISTOL MYERS SQUIBB CO (US) 1999-07-07 EP disclosed
US-5414096-A Antiviral tetrahydropyrans BRISTOL-MYERS SQUIBB CO. (US) 1995-05-09 US disclosed
EP-0608809-A1 Antiviral tetrahydropyrans BRISTOL-MYERS SQUIBB COMPANY (US) 1994-08-03 EP disclosed
US-5314893-A Antiviral tetrahydropyrans BRISTOL-MYERS SQUIBB CO. (US) 1994-05-24 US disclosed